Affinity DataIC50: 3nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of human ACAT1More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 820nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of ACAT in human J774A.1 cells assessed as reduction in esterified-cholesterol accumulation after 18 hrs in presence of 25-hydroxycholeste...More data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of human ACAT2More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 1.36E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 3.61E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 3.12E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 3.39E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 1.50E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 850nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 450nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 1.55E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 760nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 1.46E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 820nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 380nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 670nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 2.74E+3nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 400nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 560nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 650nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147](Saccharomyces bayanus (Yeast))
Kowa
US Patent
Kowa
US Patent
Affinity DataEC50: 590nMAssay Description:As an expression vector, a chimera in which DNA binding domain of Gal4, which is a yeast transcription factor, and ligand binding domain of human PPA...More data for this Ligand-Target Pair
Affinity DataEC50: 793nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 129nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 353nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair