Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetcholinergic receptor, nicotinic, alpha 1 (Muscle) isoform X1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetcholinergic receptor, nicotinic, alpha 1 (Muscle) isoform X1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetcholinergic receptor, nicotinic, alpha 1 (Muscle) isoform X1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.0200nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.0400nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Targetneuronal acetylcholine receptor subunit alpha-2(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
Targetcholinergic receptor, nicotinic, alpha 1 (Muscle) isoform X1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.0800nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
TargetCholinergic receptor nicotinic alpha 5 subunit(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.230nMAssay Description:Antagonistic activity measured for 5-hydroxytryptamine 2A receptor using [3H]-MDL- 100,907 as radioligand in rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]MDL100907 from 5HT2A receptor in Sprague-Dawley rat brain by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Affinity for cloned Y2 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Affinity for cloned Y4 receptor using [125I]-PP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of E2-Alexa633 from GFP-tagged ERalpha expressed in COS7 cells by FACSMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Agonistic activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
Targetneuronal acetylcholine receptor subunit alpha-4(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Displacement of E2-Alexa633 from GFP-tagged ERbeta expressed in COS7 cells by FACSMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [125]PYY from human chimeric NPY Y5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Agonistic activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as radioligandMore data for this Ligand-Target Pair
TargetCholinergic receptor, nicotinic alpha 1(Xenopus)
University of Miami
Curated by PDSP Ki Database
University of Miami
Curated by PDSP Ki Database
Affinity DataKi: 0.480nMAssay Description:Binding activity against cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligand.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
University Of Cincinnati And Va Medical Centers
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Affinity for cloned Y1 receptor using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
TargetVasopressin V1b receptor(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]Arg8-vasopressin from human vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2A receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 0.75nMAssay Description:Displacement of [125]PYY from human chimeric NPY Y5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Binding affinity at cloned rat 5-hydroxytryptamine 2C receptor using [3H]-DOI as radioligandMore data for this Ligand-Target Pair