TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 0.900nM ΔG°: -53.7kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 1.60nM ΔG°: -52.2kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 2nM ΔG°: -51.6kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 4.80nM ΔG°: -49.4kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 22nM ΔG°: -45.5kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 90nM ΔG°: -41.8kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 166nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 265nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 480nM ΔG°: -37.5kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 481nM ΔG°: -37.5kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Inhibition of human Thymidylate synthase (TS)More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibitory activity HIV-1 protease enzymeMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 1.10E+3nM ΔG°: -35.4kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 1.20E+3nM ΔG°: -35.2kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of Escherichia coli Thymidylate synthase (TS)More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Agouron Pharmaceuticals
Agouron Pharmaceuticals
Affinity DataKi: 1.40E+3nM ΔG°: -34.8kJ/molepH: 5.6 T: 2°CAssay Description:Protease activity was measured by continuous chromogenic assay. The chromogenic peptide His-Lys-Ala-Arg-Val-Leu- (p-NO2-Phe)-Glu-Ala-Nleu-Ser (Bache...More data for this Ligand-Target Pair