TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataKi: 250nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataKi: 1.60E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.460nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.560nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.580nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.650nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.680nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.710nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.720nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.740nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.770nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.780nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.780nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.790nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.01nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.05nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.07nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.08nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.17nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.26nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.48nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.52nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.52nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.58nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.74nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.77nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.82nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.90nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.63nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.65nMAssay Description:Displacement of [3H]SQ29,548 from TPalpha receptor (short isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.68nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3.53nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 4.43nMAssay Description:Displacement of [3H]SQ29,548 from TPbeta receptor (long isoform) expressed in COS7 cells at 1 uMMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
University of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 13.6nMAssay Description:Activity at TPbeta (long isoform) receptor expressed in HEK293 cells assessed as ability to antagonize U46619-mediated calcium ion mobilizationMore data for this Ligand-Target Pair