Compile Data Set for Download or QSAR
maximum 50k data
Found 40 with Last Name = 'porcari' and Initial = 'r'
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  3.10nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369541(CHEMBL608901)
Affinity DataIC50:  35nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369528(NSC-154020 | TRICIRIBINE)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50422306(Phosphate Salt Of Tricyclic Nucleoside | TRICIRIBI...)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369528(NSC-154020 | TRICIRIBINE)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50422306(Phosphate Salt Of Tricyclic Nucleoside | TRICIRIBI...)
Affinity DataIC50:  40nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369542(CHEMBL611850)
Affinity DataIC50:  100nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369534(CHEMBL607723)
Affinity DataIC50:  250nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369533(CHEMBL611245)
Affinity DataIC50:  350nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369536(CHEMBL611242)
Affinity DataIC50:  500nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369540(CHEMBL608301)
Affinity DataIC50:  800nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369535(CHEMBL607724)
Affinity DataIC50:  800nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369537(CHEMBL611243)
Affinity DataIC50:  1.00E+3nMAssay Description:Antiviral activity was evaluated by Reverse transcriptase activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369539(CHEMBL610949)
Affinity DataIC50:  6.80E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369532(CHEMBL610657)
Affinity DataIC50:  8.00E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369538(CHEMBL609191)
Affinity DataIC50:  8.40E+3nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063941(5,6-Dichloro-1-(4-chloro-benzyl)-1H-benzoimidazol-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase (RT) assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063977(5,6-Dichloro-1-(4-trifluoromethyl-benzyl)-1H-benzo...)
Affinity DataIC50:  2.00E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50408925(CHEMBL2112098)
Affinity DataIC50:  2.10E+4nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063948(2-Bromo-5,6-dichloro-1-(3-nitro-benzyl)-1H-benzoim...)
Affinity DataIC50: >3.20E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase (RT) assay in CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM52947((2Z,4S,4aR,5S,5aR,6R,12aS)-2-[amino(hydroxy)methyl...)
Affinity DataIC50:  4.70E+4nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM92397(4-epi-oxytetracycline)
Affinity DataIC50:  4.90E+4nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM37536((2E,4S,4aR,5S,5aR,6S,12aS)-2-[amino(hydroxy)methyl...)
Affinity DataIC50:  6.30E+4nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063945(2-Bromo-5,6-dichloro-1-(3-methyl-benzyl)-1H-benzoi...)
Affinity DataIC50:  6.60E+4nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM55038((2E,4S,4aR,5S,5aR,12aS)-2-[amino(hydroxy)methylene...)
Affinity DataIC50:  6.90E+4nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM92395(Meclocycline)
Affinity DataIC50:  9.80E+4nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369531(CHEMBL608900)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369530(CHEMBL1790617)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50089381(5-(3-Amino-5-methyl-5H-1,4,5,6,8-pentaaza-acenapht...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50089382(CHEMBL315509 | [4-(3-Amino-5-methyl-5H-1,4,5,6,8-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 Reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369543(CHEMBL610370)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was evaluated by RT (reverse transcriptase) activity in cells acutely infected with HIV-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50369527(CHEMBL609194)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50089380(CHEMBL81002 | [5-(3-Amino-5-methyl-5H-1,4,5,6,8-pe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity was tested in cells acutely infected with HIV-1 RT (reverse transcriptase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063970(2-Bromo-5,6-dichloro-1-(3,4-dichloro-benzyl)-1H-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063958(2,5,6-Trichloro-1-(4-nitro-benzyl)-1H-benzoimidazo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063972(2,5,6-Trichloro-1-(4-methyl-benzyl)-1H-benzoimidaz...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063937(2-Bromo-5,6-dichloro-1-(4-methoxy-benzyl)-1H-benzo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50063968(1-(3,5-Bis-trifluoromethyl-benzyl)-2-bromo-5,6-dic...)
Affinity DataIC50: >1.00E+5nMAssay Description:Antiviral activity against Human Immunodeficiency Virus by Reverse transcriptase assay in CEM-SS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM92398(Rolitetracycline)
Affinity DataIC50:  1.36E+5nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2-microglobulin(Homo sapiens (Human))
University of Pavia

LigandPNGBDBM92399(Anhydrochlortetracycline)
Affinity DataIC50:  1.36E+5nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild type beta-m fibrillogenesis tetracycline congeners and was follow by thioflavin fluorescence assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed