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Found 245 with Last Name = 'prasad' and Initial = 'r'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316843(2-Phenyl-4-(prop-2-yn-1-yloxy)-5,6,7,8-tetrahydro[...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316849(2-(4-Fluorobenzyl)-5,6-dimethyl-3-prop-2-yn-1-ylth...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316851(2-Phenyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316847(2,5,6-Trimethyl-3-prop-2-yn-1-ylthieno[2,3-d]pyrim...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316850(2-Methyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316845(2-Methyl-3-prop-2-yn-1-yl-5, 6, 7, 8-tetrahydro [1...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316846(2-(4-Fluorobenzyl)-3-prop-2-yn-1-yl-5,6,7,8-tetrah...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50326165(CHEMBL1241315 | oxalylaminobenzoic acid)
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant PTP1B after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316850(2-Methyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316846(2-(4-Fluorobenzyl)-3-prop-2-yn-1-yl-5,6,7,8-tetrah...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316848(5,6-Dimethyl-2-phenyl-3-prop-2-yn-1-ylthieno[2, 3-...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50326165(CHEMBL1241315 | oxalylaminobenzoic acid)
Affinity DataKi:  65nMAssay Description:Inhibition of human recombinant TCPTP after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316847(2,5,6-Trimethyl-3-prop-2-yn-1-ylthieno[2,3-d]pyrim...)
Affinity DataKi:  3.79E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50296368(7-(biphenyl-4-yl)-4-oxo-4H-chromene-3-carbaldehyde...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of human recombinant PTP1B after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50133280(5-(3-(3-(3-hydroxy-2-(methoxycarbonyl)phenoxy)prop...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of human recombinant PTP1B after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316849(2-(4-Fluorobenzyl)-5,6-dimethyl-3-prop-2-yn-1-ylth...)
Affinity DataKi:  7.62E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316851(2-Phenyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  9.70E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membrane after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50296368(7-(biphenyl-4-yl)-4-oxo-4H-chromene-3-carbaldehyde...)
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of human recombinant TCPTP after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Glenmark Research Center

Curated by ChEMBL
LigandPNGBDBM50133280(5-(3-(3-(3-hydroxy-2-(methoxycarbonyl)phenoxy)prop...)
Affinity DataKi:  2.02E+5nMAssay Description:Inhibition of human recombinant TCPTP after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057114((2-Benzooxazol-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4-...)
Affinity DataIC50:  5.25nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057102(CHEMBL10410 | [2-(2-Methanesulfonyl-2,3-dihydro-1H...)
Affinity DataIC50:  5.81nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM22416((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...)
Affinity DataIC50:  6.43nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057099(CHEMBL9970 | [2-(2,2-Dioxo-2,3-dihydro-1H-2lambda*...)
Affinity DataIC50:  6.67nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Cambridge Neuroscience

Curated by ChEMBL
LigandPNGBDBM50010747(CHEMBL543201 | CHEMBL78777 | N,N'-Bis-(3-ethyl-phe...)
Affinity DataIC50:  8nMAssay Description:Tested in vitro for the concentration required to inhibit specific [3H]-DTG radioligand binding to sigma receptor on guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057101((2-Benzothiazol-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4...)
Affinity DataIC50:  8.94nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057108(6-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50:  9.47nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057135(CHEMBL9896 | [2-(1H-Benzoimidazol-5-yl)-ethyl]-((R...)
Affinity DataIC50:  11.3nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057124(CHEMBL430314 | [2-(2,3-Dihydro-1H-isoindol-5-yl)-e...)
Affinity DataIC50:  11.6nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057098((2-Benzo[1,3]dioxol-5-yl-ethyl)-((R)-5-methoxy-1,2...)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Cambridge Neuroscience

Curated by ChEMBL
LigandPNGBDBM50010758(CHEMBL312600 | N,N'-Bis-(2-iodo-phenyl)-guanidine)
Affinity DataIC50:  13nMAssay Description:Tested in vitro for the concentration required to inhibit specific [3H]-DTG radioligand binding to sigma receptor on guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057128((2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  13.1nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Cambridge Neuroscience

Curated by ChEMBL
LigandPNGBDBM50010760(CHEMBL310170 | N,N'-Bis-(2-ethyl-phenyl)-guanidine)
Affinity DataIC50:  14nMAssay Description:Tested in vitro for the concentration required to inhibit specific [3H]-DTG radioligand binding to sigma receptor on guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057113(CHEMBL9912 | [2-(2,3-Dihydro-benzofuran-5-yl)-ethy...)
Affinity DataIC50:  14.6nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM50190682(CHEMBL3919290)
Affinity DataIC50:  15nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057110(5-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50:  16.3nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057104((2-Benzooxazol-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-...)
Affinity DataIC50:  16.7nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057142((2-Benzofuran-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-t...)
Affinity DataIC50:  17.6nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057125(CHEMBL274391 | [2-(2,3-Dihydro-benzofuran-6-yl)-et...)
Affinity DataIC50:  18.1nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057145(((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylm...)
Affinity DataIC50:  18.1nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM50190715(CHEMBL3955641)
Affinity DataIC50:  19nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM50190691(CHEMBL3935473)
Affinity DataIC50:  19nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM50190685(CHEMBL3901729)
Affinity DataIC50:  19nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057131(6-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50:  19.4nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057129((2-Indan-5-yl-ethyl)-((R)-5-methoxy-1,2,3,4-tetrah...)
Affinity DataIC50:  20.5nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Rallis India

Curated by ChEMBL
LigandPNGBDBM50190712(CHEMBL3929105)
Affinity DataIC50:  20.6nMAssay Description:Inhibition of BRC/ABL1 (unknown origin) after 40 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057093((2-Benzo[1,3]dioxol-5-yl-ethyl)-(5-methoxy-1,2,3,4...)
Affinity DataIC50:  20.6nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50057095(5-{2-[((R)-5-Methoxy-1,2,3,4-tetrahydro-naphthalen...)
Affinity DataIC50:  22.2nMAssay Description:Inhibition of uptake of [3H]-5-HT in synaptosomes from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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