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Found 55 with Last Name = 'ramajayam' and Initial = 'r'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049642(3-Chloro-4,4',5'-trifluoro-4''-methanesulfonyl-[1,...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
The M.S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50478032(CHEMBL275658 | GW4511 | GW564511 | GW69564)
Affinity DataIC50: <2nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50288291(3-(4-Methanesulfonyl-phenyl)-4,4-dimethyl-2-phenyl...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of COX-2 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50289328(5-(4-Methanesulfonyl-phenyl)-6-phenyl-2-trifluorom...)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant human COX-2 expressed in CHO-K1 cells using arachidonic acid as substrate preincubated for 15 mins followed by substrate ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50474760(CG-100649 | CG100649 | Polmacoxib)
Affinity DataIC50:  3nMAssay Description:Inhibition of COX-1 in LPS-induced mouse peritoneal macrophagesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50153982(2-(4-Ethoxy-phenyl)-3-(4-methanesulfonyl-phenyl)-p...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human COX-2 expressed in human COS cells using arachidonic acid as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50131593(4-[4-Chloro-5-(3-fluoro-4-methoxy-phenyl)-imidazol...)
Affinity DataIC50:  5nMAssay Description:Inhibition of COX-2 in human 143982 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM13063(4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)benzene-1-sul...)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049041(5-(4-Fluoro-phenyl)-6-(4-methanesulfonyl-phenyl)-s...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
The M.S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50478032(CHEMBL275658 | GW4511 | GW564511 | GW69564)
Affinity DataIC50: <10nMAssay Description:Inhibition of HIV1 reverse transcriptase Y181C mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
The M.S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50478032(CHEMBL275658 | GW4511 | GW564511 | GW69564)
Affinity DataIC50: <10nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50507137(CHEMBL4533150)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50102311(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-6...)
Affinity DataIC50:  12nMAssay Description:Inhibition of COX-2 in human 143982 cells using arachidonic acid as substrate preincubated for 15 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50029600(5-Bromo-2-(4-fluoro-phenyl)-3-(4-methanesulfonyl-p...)
Affinity DataIC50:  14nMAssay Description:Inhibition of COX-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50289303(5-(4-Methanesulfonyl-phenyl)-6-phenyl-3,5-dihydro-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human COX-2 transfected in CHO cells using arachidonic acid as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50507138(CHEMBL4473838)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049026(5-(4-Fluoro-phenyl)-6-(4-methanesulfonyl-phenyl)-s...)
Affinity DataIC50:  26nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50029614((SC-57666)1-[2-(4-fluorophenyl)-1-cyclopentenyl]-4...)
Affinity DataIC50:  26nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50103314(4-(4-Fluoro-phenyl)-5-(4-methanesulfonyl-phenyl)-2...)
Affinity DataIC50:  32nMAssay Description:Inhibition of ovine COX-2 using arachidonic acid as substrate by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50076873(2-(2-Chloro-phenyl)-4-(4-fluoro-phenyl)-5-(4-metha...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human COX-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50286048(2-Bromo-3-(4-fluoro-phenyl)-4-(4-methanesulfonyl-p...)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50286048(2-Bromo-3-(4-fluoro-phenyl)-4-(4-methanesulfonyl-p...)
Affinity DataIC50:  80nMAssay Description:Inhibition of COX-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50072064(5-Chloro-3-(4-methanesulfonyl-phenyl)-6''-methyl-[...)
Affinity DataIC50:  81nMAssay Description:Inhibition of human COX-2 transfected in CHO cells using arachidonic acid as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50125624(3-(4-Chloro-phenyl)-5-hydroxy-4-(4-methanesulfonyl...)
Affinity DataIC50:  110nMAssay Description:Inhibition of COX-2 (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50091181(4-[2-(4-Methyl-thiazol-2-yl)-4-trifluoromethyl-imi...)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50103510(4-(4-Azido-phenyl)-3-phenyl-5H-furan-2-one | CHEMB...)
Affinity DataIC50:  196nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM22369(4-(4-methanesulfonylphenyl)-3-phenyl-2,5-dihydrofu...)
Affinity DataIC50:  500nMAssay Description:Inhibition of COX-2 in human whole bloodMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50075664(2-(3,5-Difluoro-phenyl)-3-(4-methanesulfonyl-pheny...)
Affinity DataIC50:  620nMAssay Description:Inhibition of COX-2 in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50150218(3-(4-Fluoro-phenoxy)-2-(4-methanesulfonyl-phenyl)-...)
Affinity DataIC50:  980nMAssay Description:Inhibition of COX-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50129503(6-Ethoxy-3-(4-methanesulfonyl-phenyl)-4-phenyl-pyr...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of ovine COX-2 using arachidonic acid as substrate preincubated for 2 mins followed by substrate addition and measured after 2 mins by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50084361(4-[3-(4-Fluoro-phenyl)-2-oxo-2,3-dihydro-oxazol-4-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of COX-2 in LPS-stimulated human whole blood after 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50103509(1-(4-Azido-phenyl)-5-p-tolyl-3-trifluoromethyl-1H-...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50091171(3-[1-(4-Methanesulfonyl-phenyl)-4-trifluoromethyl-...)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483060(CHEMBL1277046 | acs.jmedchem.1c00409_ST.374)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483064(CHEMBL1277227)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483065(CHEMBL1277228)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483065(CHEMBL1277228)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The M.S University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50057877(4-[2-(4-Fluoro-phenyl)-pyrrol-1-yl]-benzenesulfona...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of recombinant human COX-2 expressed in Baculovirus infected sf9 cells using arachidonic acid as substrate preincubated for 10 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483062(CHEMBL1277135)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483059(CHEMBL1276871)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483058(CHEMBL1278125)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483059(CHEMBL1276871)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483062(CHEMBL1277135)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483057(CHEMBL1277944)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483060(CHEMBL1277046 | acs.jmedchem.1c00409_ST.374)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
The M.S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50470153(CHEMBL415908)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483064(CHEMBL1277227)
Affinity DataIC50:  2.24E+4nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483063(CHEMBL1277136)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of SARS coronavirus 3C-like protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Coxsackievirus B3 (strain Nancy))
Academia Sinica

Curated by ChEMBL
LigandPNGBDBM50483058(CHEMBL1278125)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of coxsackievirus B3 3C protease by fluorescence plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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