Compile Data Set for Download or QSAR
maximum 50k data
Found 424 with Last Name = 'ramunno' and Initial = 'a'
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118528(CHEMBL135514 | Ethyl-carbamic acid 5-phenyl-6-oxa-...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]-Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118528(CHEMBL135514 | Ethyl-carbamic acid 5-phenyl-6-oxa-...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118537(CHEMBL135391 | Ethyl-carbamic acid 7-chloro-5-phen...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118528(CHEMBL135514 | Ethyl-carbamic acid 5-phenyl-6-oxa-...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]-PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118539(CHEMBL136036 | Diethyl-carbamic acid 5-thiophen-2-...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118541(CHEMBL445583 | Cyclopropyl-carbamic acid 5-phenyl-...)
Affinity DataKi:  0.310nMAssay Description:Inhibition of [3H]-PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118534(CHEMBL136926 | Dimethyl-carbamic acid 5-p-tolyl-6-...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118541(CHEMBL445583 | Cyclopropyl-carbamic acid 5-phenyl-...)
Affinity DataKi:  0.470nMAssay Description:Inhibition of [3H]-Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50100706(2-Bromo-5-(1-methyl-pyrrolidin-2-yl)-pyridine | CH...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118542(CHEMBL335300 | Diethyl-carbamic acid 5-m-tolyl-6-o...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50078056(2-Chloro-5-(1-methyl-pyrrolidin-2-yl)-pyridine | C...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118545(CHEMBL133144 | Ethyl-carbamic acid 5-p-tolyl-6-oxa...)
Affinity DataKi:  0.680nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118544(CHEMBL335085 | Methyl-propyl-carbamic acid 5-pheny...)
Affinity DataKi:  0.690nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118527(CHEMBL336774 | Methyl-carbamic acid 5-phenyl-6-oxa...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of [3H]-Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118543(CHEMBL341455 | Ethyl-methyl-carbamic acid 5-phenyl...)
Affinity DataKi:  0.780nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118535(CHEMBL135801 | Propyl-carbamic acid 5-phenyl-6-oxa...)
Affinity DataKi:  0.910nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118529(Butyl-methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118527(CHEMBL336774 | Methyl-carbamic acid 5-phenyl-6-oxa...)
Affinity DataKi:  0.960nMAssay Description:Inhibition of [3H]-PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118546(CHEMBL134781 | Diethyl-carbamic acid 5-m-tolyl-6-o...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118547(CHEMBL135428 | Diethyl-carbamic acid 5-(3,5-difluo...)
Affinity DataKi:  1.26nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118531(CHEMBL135327 | Diethyl-carbamic acid 5-phenyl-6-ox...)
Affinity DataKi:  1.77nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474925(CHEMBL294757)
Affinity DataKi:  1.80nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474925(CHEMBL294757)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50475399(CHEMBL364003 | US10667515, Compound 5-methyl-nicot...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50475402(CHEMBL382287)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118541(CHEMBL445583 | Cyclopropyl-carbamic acid 5-phenyl-...)
Affinity DataKi:  2.21nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118527(CHEMBL336774 | Methyl-carbamic acid 5-phenyl-6-oxa...)
Affinity DataKi:  2.26nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM21279(1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118540(Acetic acid 5-m-tolyl-6-oxa-10b-aza-benzo[e]azulen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]-Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50052594((+) 3-Bromo-5-(1-methyl-pyrrolidin-2-yl)-pyridine ...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474921(CHEMBL103225)
Affinity DataKi:  5.60nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118533(CHEMBL336903 | Diethyl-carbamic acid 5-phenyl-6H-b...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]-PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  6.03nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50052594((+) 3-Bromo-5-(1-methyl-pyrrolidin-2-yl)-pyridine ...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50052594((+) 3-Bromo-5-(1-methyl-pyrrolidin-2-yl)-pyridine ...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118536(4-Methyl-piperazine-1-carboxylic acid 5-phenyl-6-o...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102265(1-(5-Bromo-pyridin-2-yl)-3-[2-(6-fluoro-4-oxo-4H-p...)
Affinity DataKi:  9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50102271(1-(5-Bromo-pyridin-2-yl)-3-[2-(4-oxo-4H-5,9,9b-tri...)
Affinity DataKi:  9nMAssay Description:Inhibition of HIV-1 wild-type RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  10nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution V106AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474922(CHEMBL190652)
Affinity DataKi:  10nMAssay Description:Binding affinity for rat brain Nicotinic acetylcholine receptor alpha4-beta2 using [3H]S-(-)-nicotineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474922(CHEMBL190652)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118531(CHEMBL135327 | Diethyl-carbamic acid 5-phenyl-6-ox...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]-PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universita' Degli Studi Di Salerno

Curated by ChEMBL
LigandPNGBDBM50082061((+/-)-5-ethyl-5-(3-methoxy-phenyl)-6-oxa-10b-aza-b...)
Affinity DataKi:  11nMAssay Description:In vitro inhibitory activity of the compound against HIV-1 mutant Reverse transcriptase containing the single amino acid substitution L100IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50118538(CHEMBL135663 | Diethyl-carbamic acid 5-thiophen-2-...)
Affinity DataKi:  11.5nMAssay Description:Inhibition of [3H]-PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 424 total ) | Next | Last >>
Jump to: