Affinity DataKi: 3.08E+4nMAssay Description:Inhibition of cathepsin D in human liver using Lys-Lys-Pro-Ala-Glu-Phe-Phe-Ala-Leu-Lys as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Inhibition of cathepsin D in human liver using Lys-Lys-Pro-Ala-Glu-Phe-Phe-Ala-Leu-Lys as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+5nMAssay Description:Non-competitive inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using varying levels...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+5nMAssay Description:Non-competitive inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using varying levels...More data for this Ligand-Target Pair
Affinity DataKi: 4.16E+5nMAssay Description:Inhibition of recombinant BACE-1 (unknown origin) expressed in Escherichia coli measured for 5 to 30 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.16E+5nMAssay Description:Inhibition of recombinant BACE-1 (unknown origin) expressed in Escherichia coli measured for 5 to 30 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+5nMAssay Description:Non-competitive inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using varying levels...More data for this Ligand-Target Pair
Affinity DataKi: 7.30E+6nMAssay Description:Inhibition of Trypanosoma cruzi trans-sialidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+7nMAssay Description:Inhibition of recombinant Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate after 10 mins in prese...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of Trypanosoma cruzi trans-sialidase using CF3MuSA as substrate by UV/visible spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+5nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+6nMAssay Description:Inhibition of Streptococcus pneumoniae neuraminidase A using MuNANA as substrate pretreated for 10 mins followed by substrate addition by fluorescenc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+6nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: 2.39E+6nMAssay Description:Inhibition of Clostridium perfringens neuraminidase using MuNANA as substrate pretreated for 10 mins followed by substrate addition by fluorescence a...More data for this Ligand-Target Pair
Affinity DataIC50: 5.58E+6nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataIC50: >7.50E+6nMAssay Description:Inhibition of recombinant HisA-tagged Trypanosoma cruzi trans-sialidase expressed in Escherichia coli BL21 (DE3) using MuNANA as substrate pretreated...More data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+4nMAssay Description:Inhibition of BACE-1 in CHO cells expressing wild-type APP assessed as reduction in amyloid beta-40 production after 6 hrs by sandwich ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 2.17E+5nMAssay Description:Inhibition of BACE-1 in human SH-SY5Y cells expressing wild-type APP assessed as reduction in amyloid beta-40 production after 16 hrs by sandwich ELI...More data for this Ligand-Target Pair