Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor measured by displacing [3H]-8-OH-DPAT from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.11nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine receptor D2 from rat striatumMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.64nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine receptor D2 from rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor measured by displacing [3H]-prazosin from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16.1nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 16.9nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 19.1nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine receptor D2 from rat striatumMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22.4nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 24.0nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:In vitro binding affinity at human Alpha-1D adrenergic receptor.More data for this Ligand-Target Pair
Affinity DataKi: 27.8nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine receptor D2 from rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 31.1nMAssay Description:In vitro binding affinity at human Alpha-1B adrenergic receptor.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 35.0nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity at human Alpha-1A adrenergic receptor.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor measured by displacing [3H]-8-OH-DPAT from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 64.9nMAssay Description:Binding affinity to 5HT1AMore data for this Ligand-Target Pair
Affinity DataKi: 83.0nMAssay Description:Inhibtion of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor from rat hippocampusMore data for this Ligand-Target Pair