TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
Affinity DataKi: 9.20E+4nMAssay Description:Compound was tested for inhibitory activity against recombinant Trypanothione reductase from Trypanosoma cruziMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against opioid receptor sigma 1 of guinea pig cerebral cortex using [3H]-(+)-pentazocine upon incubation for 150 minutes at ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration against opioid receptor sigma 1 of guinea pig cerebral cortex using [3H]-(+)-pentazocine upon incubation for 150 minutes at ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMpH: 7.5 T: 2°CAssay Description:Inhibitory activity against Opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 microM in LLCPKI cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibitory concentration against opioid receptor sigma 1 of guinea pig cerebral cortex using [3H]-(+)-pentazocine upon incubation for 150 minutes at ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:In vitro inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 microM in LLCPKI cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10.5nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 11.7nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 13.6nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory concentration against opioid receptor sigma 1 of guinea pig cerebral cortex using [3H]-(+)-pentazocine upon incubation for 150 minutes at ...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 21.5nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair
Affinity DataIC50: 21.5nMAssay Description:Inhibitory concentration against opioid receptor sigma 1 of guinea pig cerebral cortex using [3H]-(+)-pentazocine upon incubation for 150 minutes at ...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of Prolyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 23.3nMAssay Description:In vitro inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 23.5nMAssay Description:In vitro inhibition of beta-hematin formationMore data for this Ligand-Target Pair
Affinity DataIC50: 23.8nMpH: 7.5Assay Description:Inhibitory activity against opioid receptor sigma 1 in guinea pig cerebral cortex using [3H]-(+)-pentazocine as radio ligand at pH 7.5 for 150 min at...More data for this Ligand-Target Pair