Affinity DataKi: 0.430nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Ability of the compound to reverse Neuropeptide Y receptor type 1-induced inhibition of forskolin-induced inhibition of forskolin-stimulated cAMPMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of [3H]-AMPA binding to human GluR2 receptors expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 287nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 442nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Binding affinity to GluK1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 522nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
Affinity DataKi: 559nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 565nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 743nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Binding affinity to GluK1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Binding affinity to GluK1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 915nMAssay Description:Inhibition of [3H]spiperone binding to Dopamine receptor D2 at 0.02 nMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair