Affinity DataKi: 0.140nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Displacement of [125I]CXCL10 from human CXCR3 expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity was evaluated against thymidylate synthaseMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:The compound was evaluated in vitro for the thrombin inhibition.More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:The compound was evaluated in vitro for the thrombin inhibition.More data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity was evaluated against dihydrofolate reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 15.8nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Histamine H3 receptor competition binding using [3H]Na-methylhistamineMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Displacement of [125I]-CXCL10 from human CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Pharmacopeia Drug Discovery
Curated by ChEMBL
Pharmacopeia Drug Discovery
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to human CXCR2 receptor transfected in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Displacement of [125I]CXCL10 from CXCR3 expressed in HEK293 cellsMore data for this Ligand-Target Pair