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Found 242 with Last Name = 'soca' and Initial = 'l'
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296089(2-(2-(5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)ben...)
Affinity DataIC50:  0.910nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296106(3-(5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296115(3-(5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296095(2-(2-(1H-tetrazol-5-yl)ethyl)-9-(3-(2-(7-chloroqui...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296092(3-(5-(3-((7-chloroquinolin-2-yl)ethynyl)benzyl)-3,...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296105(3-(5-(3-(2-(7-chloro-6-fluoroquinolin-2-yl)vinyl)b...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296114(3-(5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296088(4-((5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)benzy...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296085(2-(1-((5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296103(3-(5-(3-(2-(7-fluoroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  3.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296102(4-(1-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-2-...)
Affinity DataIC50:  3.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296087(4-(5-(3-((E)-2-(7-chloroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  4.10nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296101(4-(1-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-1H...)
Affinity DataIC50:  4.40nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296113(3-(5-(3-(2-(6,7-difluoroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296099(3-(9-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-9H...)
Affinity DataIC50:  4.80nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296100(2-(9-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-2,...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296112(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-8-...)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296097(3-((2-(1-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  9.30nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296096(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296116(3-(5-((2-(7-chloroquinolin-2-yl)benzofuran-5-yl)me...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296094(4-(9-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-4,...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296081(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296111(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-7-...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296084(5-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296082(2-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296093(3-(9-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-4,...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296104(3-(5-(3-(2-(6,7-dichloroquinolin-2-yl)vinyl)benzyl...)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296091(3-(5-(3-(2-(7-chloroquinolin-2-yl)ethyl)benzyl)-3,...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296086(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296083(4-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-3,...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296107(3-(5-(3-(2-(4-tert-butylthiazol-2-yl)vinyl)benzyl)...)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296090(3-(5-(3-((7-chloroquinolin-2-yl)methoxy)benzyl)-3,...)
Affinity DataIC50:  42nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296109(3-(5-(3-(2-(2,3-dichlorothieno[3,2-b]pyridin-5-yl)...)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150210(3-(2-Fluoro-4-methyl-phenoxy)-2-(4-methanesulfonyl...)
Affinity DataIC50:  60nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296098(3-(((1-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-...)
Affinity DataIC50:  61nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150211(3-(2,4-Difluoro-phenoxy)-2-(4-methanesulfonyl-phen...)
Affinity DataIC50:  80nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296108(3-(5-(3-(2-(5-chlorobenzo[d]thiazol-2-yl)vinyl)ben...)
Affinity DataIC50:  112nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50296110(3-(5-(3-(2-(7-chloroquinolin-2-yl)vinyl)benzyl)-6-...)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]LTD4 from CYSLT1 receptor in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150226(3-(4-Bromo-2-fluoro-phenoxy)-2-(4-methanesulfonyl-...)
Affinity DataIC50:  150nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150202(2-(4-Methanesulfonyl-phenyl)-6-methyl-3-o-tolyloxy...)
Affinity DataIC50:  170nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150193(3-(2-Chloro-4-methoxy-phenoxy)-2-(4-methanesulfony...)
Affinity DataIC50:  180nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150215(3-(4-Fluoro-2-methyl-phenoxy)-2-(4-methanesulfonyl...)
Affinity DataIC50:  180nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150197(3-(4-Chloro-2-methyl-phenoxy)-2-(4-methanesulfonyl...)
Affinity DataIC50:  190nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(RAT)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory concentration against rat prostaglandin G/H synthase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150185(3-(4-Chloro-2-fluoro-phenoxy)-2-(4-methanesulfonyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50150224(2-(4-Methanesulfonyl-phenyl)-6-methyl-3-p-tolyloxy...)
Affinity DataIC50:  210nMAssay Description:Inhibition concentration against cyclooxygenase-2 (COX-2) in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50084355(4-[3-(4-Methoxy-phenyl)-2-oxo-2,3-dihydro-oxazol-4...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against prostaglandin G/H synthase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(RAT)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50105290(2-[7-Methoxy-4-(4-methyl-benzyl)-naphthalen-1-yl]-...)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration against rat Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against prostaglandin G/H synthase 2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(RAT)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration against rat Prostaglandin G/H synthase 2More data for this Ligand-Target Pair
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