Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 0.380nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to rat cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 14.9nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 17.4nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 31.4nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 63.2nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 72.1nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Displacement of [3H]LSD from rat rat kidney proximal convoluted tubule 5HT7R expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 243nMAssay Description:Displacement of [3H]LSD from rat rat kidney proximal convoluted tubule 5HT7R expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 352nMAssay Description:Displacement of [3H]LSD from rat rat kidney proximal convoluted tubule 5HT7R expressed in COS7 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataKi: 476nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]-5-CT from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 438nMAssay Description:Antagonist activity at human 5HT7A receptor expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP accumulation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 531nMAssay Description:Antagonist activity at human 5HT7A receptor expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP accumulation by ELISAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 21nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.324nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 3.39E+3nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 3.5nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 170nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Karolinska Institute And Karolinska University Hospital
Curated by ChEMBL
Affinity DataEC50: 0.776nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...More data for this Ligand-Target Pair