Affinity DataKi: 0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])-phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from human GPR40 receptor expressed in C...More data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptide (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from rat GPR40 receptor expressed in CHO ...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(RAT)
Takeda Chemical Industries
Curated by PDSP Ki Database
Takeda Chemical Industries
Curated by PDSP Ki Database
Affinity DataKi: 8.80nMAssay Description:Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])-phenylmethoxy]biphenyl-3-yl}methoxy)phenyl]propanoic acid from human GPR40 expressed in CHO cells a...More data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1A domain peptide (unknown origin)More data for this Ligand-Target Pair