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Found 32 with Last Name = 'szallasi' and Initial = 'a'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.0200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.0540nMAssay Description:Inhibitory constant for RTX binding to rat spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.120nMAssay Description:Inhibitory constant for RTX binding to porcine spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052327(6-hydroxy-15-isopropenyl-4,13,17-trimethyl-5-oxo-(...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  0.450nMAssay Description:Inhibitory constant for RTX binding to human spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052320(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  1nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052323((4-Hydroxy-3-methoxy-phenyl)-acetic acid 4a,7b-dih...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052333(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052328(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50196337(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataKi: <10nMAssay Description:Agonistic activity against vanilloid receptor 1 (TRPV1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052330(13-benzyl-5,6-dihydroxy-15-isopropenyl-4,17-dimeth...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052437(4-Azido-benzoic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9a...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052439((4-Azido-phenyl)-acetic acid (1aR,1bS,4aR,7aS,7bS,...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052443(CHEMBL320485 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052445(Benzoic acid (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9a-ac...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052441(CHEMBL317025 | Cyclohexyl-acetic acid (1aR,1bS,4aR...)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]RTX binding from Vanilloid receptor of rat dorsal Root Ganglion (DRG) membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052321(CHEMBL98634 | Phenyl-acetic acid (1aR,1bS,4aR,7aS,...)
Affinity DataKi:  600nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052447(CHEMBL322621 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052446(CHEMBL319644 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]- RTX binding to vanilloid receptor of rat urinary bladderMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from pig spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052448(CHEMBL107248 | Cyclohexanecarboxylic acid (1aR,1bS...)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50052440(CHEMBL104647 | Phenyl-acetic acid (1aR,1bS,4aR,7aS...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibition of [3H]- RTX binding to Vanilloid receptors from human spinal cordMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052438(CHEMBL320175 | Phenyl-acetic acid (1aR,1bS,4aR,5S,...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052324(13-benzyl-6-hydroxy-8-hydroxymethyl-15-isopropenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute

Curated by ChEMBL
LigandPNGBDBM50052444((4-Hydroxy-3-methoxy-phenyl)-acetic acid (1aR,1bS,...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]RTX from Vanilloid receptor in Rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed