TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by PDSP Ki Database
Meiji Seika Kaisha
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human FBaseMore data for this Ligand-Target Pair
Affinity DataIC50: 16.1nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human NAMPT assessed as decrease in NMN production by fluorescence based analysisMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 67.9nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Nagasaki University
Curated by ChEMBL
Nagasaki University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of eIF4A-mediated cap-dependent protein synthesis in FF-HCV-Ren mRNA transfected Swiss mouse Krebs2 cell extract by [35S]methionine metabo...More data for this Ligand-Target Pair