TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 12.4nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human PIM1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of human GST fused Pim2 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human PIM1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human PIM1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human PIM1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair