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Found 47 with Last Name = 'uchida' and Initial = 't'
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Yamanashi Medical University

Curated by ChEMBL
LigandPNGBDBM50485606(CHEBI:63925 | Latanoprost acid)
Affinity DataKi:  149nMAssay Description:TP_TRANSPORTER: inhibition of PGE1 uptake (PGE1: 0.0004 uM) in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Yamanashi Medical University

Curated by ChEMBL
LigandPNGBDBM50240648(LATANOPROST (FREE ACID) | PhXA 41 | Xalatan | isop...)
Affinity DataKi: >1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of PGE1 uptake (PGE1: 0.0004 uM) in PGT-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141316(US8653304, 3)
Affinity DataIC50:  3nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141323(US8653304, 108b)
Affinity DataIC50:  13nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141317(US8653304, 46b | US8653304, 47b)
Affinity DataIC50:  15nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141321(US8653304, 84b)
Affinity DataIC50:  16nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141317(US8653304, 46b | US8653304, 47b)
Affinity DataIC50:  18nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141320(US8653304, 52b)
Affinity DataIC50:  24nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141324(US8653304, 123b)
Affinity DataIC50:  29nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141319(US8653304, 50b)
Affinity DataIC50:  35nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141322(US8653304, 92b)
Affinity DataIC50:  51nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Toray Industries

US Patent
LigandPNGBDBM141325(US8653304, Comparative Compound 1)
Affinity DataIC50:  117nMT: 2°CAssay Description:Using human p38 MAPK alpha , the p38 MAPK inhibitory activity of Compound (I) was studied by a method partially modified from the method described in...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53408((2S)-2-[[5-(3,4-dihydro-1H-isoquinoline-2-carbonyl...)
Affinity DataIC50: >1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53402((3R,3aR,7aR)-2-benzyl-3-(1-bromo-2-naphthyl)-7a-me...)
Affinity DataIC50:  1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012280(CHEMBL3260030)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53401((3R,3aS,7R,7aS)-2-benzyl-3-(3-chloro-4-methoxy-phe...)
Affinity DataIC50:  2.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53412(4-[[5-[[(1S)-1-tert-butoxycarbonyl-5-(tert-butoxyc...)
Affinity DataIC50:  2.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012323(CHEMBL3260378)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53403((3R,3aR,7aR)-2-benzyl-3-(5-bromo-2-methoxy-phenyl)...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53405(4-(4-methoxyphenyl)-5,8-dimethyl-2-phenyl-3,4-dihy...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53404((3R,3aR,7aR)-2-benzyl-3-[4-fluoro-3-(4-methylpheny...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012321(CHEMBL3260377)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012320(CHEMBL3260376)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM16415((1,3-dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)acetic...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53406((6Z)-1-benzoyl-4-(4-fluorobenzyl)-5-(4-methoxyphen...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53407(2-(2-methoxyphenyl)-8-nitro-5-oxidanyl-chromen-4-o...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53411((2S)-2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imida...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53410(4-[[5-[[(1S)-1-benzyl-2-tert-butoxy-2-keto-ethyl]c...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53409((2S)-2-[[4-[[(1S)-2-tert-butoxy-2-keto-1-methyl-et...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012283(CHEMBL3260369)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012286(CHEMBL3260372)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012282(CHEMBL3260368)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012284(CHEMBL3260370)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012285(CHEMBL3260371)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012288(CHEMBL3260374)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012281(CHEMBL3260031)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012289(CHEMBL3260375)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012287(CHEMBL3260373)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Japan Science And Technology Agency

Curated by ChEMBL
LigandPNGBDBM50012280(CHEMBL3260030)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Vaccinia H1-related phosphatase (unknown origin) by fluorescence emission assay in presence of 0.001% NP-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Iwate University

Curated by ChEMBL
LigandPNGBDBM50465052(CHEMBL4288015)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of human GSK-3beta using peptide substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeme oxygenase HutZ [D132E](Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  4.10E+3nMpH: 6.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme-binding protein HutZ(Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  130nMpH: 6.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme oxygenase HutZ [D132E](Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  27nMpH: 8.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme oxygenase HutZ [D132N](Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  150nMpH: 8.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme oxygenase HutZ [D132L](Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  470nMpH: 8.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme-binding protein HutZ(Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  52nMpH: 8.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme oxygenase HutZ [D132N](Vibrio cholerae)
Hokkaido University

LigandPNGBDBM231681(Hemin)
Affinity DataKd:  1.90E+3nMpH: 6.0Assay Description:Heme binding was tracked by difference spectroscopy in the Soret region of the UV−visible spectrum. Successive aliquots of 0.5 mM hemin in 0.1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed