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Found 136 with Last Name = 'van' and Initial = 'mv'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  59.8nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  169nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  973nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  1.53E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548364(WO2022093856, Example 1-59)
Affinity DataIC50:  10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataIC50:  15.7nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548305(WO2022093856, Example 1-2)
Affinity DataIC50:  19nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548347(WO2022093856, Example 1-42)
Affinity DataIC50:  22nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548341(WO2022093856, Example 1-36)
Affinity DataIC50:  23nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548358(WO2022093856, Example 1-53)
Affinity DataIC50:  24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278373(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548357(WO2022093856, Example 1-52)
Affinity DataIC50:  39nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278305(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  46nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548359(WO2022093856, Example 1-54)
Affinity DataIC50:  49nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548356(WO2022093856, Example 1-51)
Affinity DataIC50:  50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278071(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  52nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548353(WO2022093856, Example 1-48)
Affinity DataIC50:  53nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298593((R)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548360(WO2022093856, Example 1-55)
Affinity DataIC50:  57nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548337(WO2022093856, Example 1-32)
Affinity DataIC50:  57nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548334(WO2022093856, Example 1-29)
Affinity DataIC50:  57nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548343(WO2022093856, Example 1-38)
Affinity DataIC50:  60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278817(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  83nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548345(WO2022093856, Example 1-40)
Affinity DataIC50:  84nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548323(WO2022093856, Example 1-20)
Affinity DataIC50:  84nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278072(2-(R,S)-{2-[(1-Methyl-1H-indole-2-carbonyl)-amino]...)
Affinity DataIC50:  92nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548354(WO2022093856, Example 1-49)
Affinity DataIC50:  93nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298576((R)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-phe...)
Affinity DataIC50:  106nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360274(CHEMBL1933101)
Affinity DataIC50:  107nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548348(WO2022093856, Example 1-43)
Affinity DataIC50:  121nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548340(WO2022093856, Example 1-35)
Affinity DataIC50:  142nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298589((R)-2-(2-(5-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  151nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298592((+/-)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  159nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548351(WO2022093856, Example 1-46)
Affinity DataIC50:  162nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548331(WO2022093856, Example 1-26)
Affinity DataIC50:  180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548333(WO2022093856, Example 1-28)
Affinity DataIC50:  196nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548306(WO2022093856, Example 1-3)
Affinity DataIC50:  216nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGTPase KRas [1-169,G12C,C118A](Homo sapiens (Human))
Amgen

WIPO
LigandPNGBDBM548335(WO2022093856, Example 1-30)
Affinity DataIC50:  265nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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