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Found 45 with Last Name = 'westaway' and Initial = 'j'
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  10nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136494(8-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  22nMAssay Description:Binding affinity at 5-hydroxytryptamine 2A receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  70nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi:  140nMAssay Description:Binding affinity at alpha 2B adrenergic receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130262(2,3,4,9-Tetrahydro-1H-beta-carboline | CHEMBL26923...)
Affinity DataKi:  180nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136504(5-Bromo-4,9-dihydro-3H-beta-carboline | CHEMBL2675...)
Affinity DataKi:  180nMAssay Description:Binding affinity at 5-hydroxytryptamine 2A receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  330nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136501(5-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  390nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50130095(6-Methyl-1,2,3,4,5,6-hexahydro-azepino[4,5-b]indol...)
Affinity DataKi:  415nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136494(8-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  460nMAssay Description:Binding affinity at alpha-2 adrenergic receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50108307(1,2,3,4-Tetrahydro-pyrazino[1,2-a]indole | CHEMBL6...)
Affinity DataKi:  516nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM73071(2,3,4,5-tetrahydro-1H-pyrid[4,3-b]indole;hydrochlo...)
Affinity DataKi:  600nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136502(8-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi:  640nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136506(4,9-Dihydro-3H-beta-carboline | CHEMBL266221)
Affinity DataKi:  700nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50130262(2,3,4,9-Tetrahydro-1H-beta-carboline | CHEMBL26923...)
Affinity DataKi:  710nMAssay Description:Binding affinity for rat alpha-2 adrenergic receptor from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136503(8-Bromo-4,9-dihydro-3H-beta-carboline | CHEMBL6746)
Affinity DataKi:  815nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136499(5-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi:  825nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity at 5-hydroxytryptamine 2A receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223742(CHEMBL267399)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50130262(2,3,4,9-Tetrahydro-1H-beta-carboline | CHEMBL26923...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50130262(2,3,4,9-Tetrahydro-1H-beta-carboline | CHEMBL26923...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136505(6-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL67...)
Affinity DataKi:  2.19E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136504(5-Bromo-4,9-dihydro-3H-beta-carboline | CHEMBL2675...)
Affinity DataKi:  3.16E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136494(8-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  3.74E+3nMAssay Description:Binding affinity at imidazoline receptor I-1 of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50130262(2,3,4,9-Tetrahydro-1H-beta-carboline | CHEMBL26923...)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity for rat alpha-2 adrenergic receptor from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50108311(7-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  4.51E+3nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136509(8-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL26...)
Affinity DataKi:  5.02E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136508(6-Bromo-4,9-dihydro-3H-beta-carboline | CHEMBL6626)
Affinity DataKi:  5.29E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  7.41E+3nMAssay Description:Binding affinity for rat alpha-2 adrenergic receptor from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136492(6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | 6...)
Affinity DataKi:  7.83E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi:  8.84E+3nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi:  8.84E+3nMAssay Description:Binding affinity for rat alpha-2 adrenergic receptor from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50108316(8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  9.55E+3nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50108316(8-Methoxy-1,2,3,4-tetrahydro-pyrazino[1,2-a]indole...)
Affinity DataKi:  9.93E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A serotonin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079903(7-Methoxy-4,9-dihydro-3H-beta-carboline | CGS-1928...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136497(7-Bromo-4,9-dihydro-3H-beta-carboline | CHEMBL4289...)
Affinity DataKi:  1.07E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136495(6-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  1.15E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50108305(1,2,3,4-Tetrahydro-benzo[4,5]imidazo[1,2-a]pyrazin...)
Affinity DataKi:  1.34E+4nMAssay Description:Displacement of [3H]RX-821002 from alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223899(CHEBI:65009 | CHEMBL6509)
Affinity DataKi:  1.47E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136507(7-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  1.55E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50024210(1H-indole-3-ethanamine | 2-(1H-indol-3-yl)ethanami...)
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50132097(7-Methoxy-2,3,4,9-tetrahydro-1H-beta-carboline | C...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity at imidazoline receptor I-1 of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed