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Found 126 with Last Name = 'yamano' and Initial = 'm'
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0970nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPromotilin(RABBIT)
Sanwa Kagaku Kenkyusho

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPromotilin(RABBIT)
Sanwa Kagaku Kenkyusho

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Sanwa Kagaku Kenkyusho

Curated by PDSP Ki Database
LigandPNGBDBM85615(L-Phe-L-Val-L-Pro-L-Ile-L-Phe-L-Thr-L-Tyr-Gly-L-Gl...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Sanwa Kagaku Kenkyusho

Curated by PDSP Ki Database
LigandPNGBDBM85615(L-Phe-L-Val-L-Pro-L-Ile-L-Phe-L-Thr-L-Tyr-Gly-L-Gl...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82480(YM022 S-isomer)
Affinity DataKi:  140nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82480(YM022 S-isomer)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  5.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)
Affinity DataKi:  6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM25041(N'-[(1E)-{6-cyanoimidazo[1,2-a]pyridin-3-yl}methyl...)
Affinity DataIC50:  0.260nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25036(CHEMBL393525 | N'-[(1E)-{6-bromoimidazo[1,2-a]pyri...)
Affinity DataIC50:  0.300nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25037(N'-[(1E)-{6-chloroimidazo[1,2-a]pyridin-3-yl}methy...)
Affinity DataIC50:  0.770nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25052(3-{6-bromoimidazo[1,2-a]pyridin-3-yl}-1-[(2-methyl...)
Affinity DataIC50:  1.80nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25018(3-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phe...)
Affinity DataIC50:  2.5nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25018(3-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phe...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25050(3-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-1-...)
Affinity DataIC50:  2.80nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25056(4-{6-chloroimidazo[1,2-a]pyridin-3-yl}-2-[(2-methy...)
Affinity DataIC50:  2.80nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  3nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25030(3-{6-bromo-2-methylimidazo[1,2-a]pyridin-3-yl}-1-[...)
Affinity DataIC50:  3.10nMpH: 7.4 T: 2°CAssay Description:The test compounds and enzyme were mixed in buffer, and the substrate and [gamma-33P] ATP/ATP were added to the mixture to initiate the reaction. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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