TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Target4,4'-diapophytoene synthase(Staphylococcus aureus)
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition of Staphylococcus aureus dehydrosqualene synthase expressed in Escherichia coli BL21 (DE3) cells by continuous spectrophotometric assayMore data for this Ligand-Target Pair
Target4,4'-diapophytoene synthase(Staphylococcus aureus)
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of Staphylococcus aureus dehydrosqualene synthase expressed in Escherichia coli BL21 (DE3) cells by continuous spectrophotometric assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Antagonist activity at full length recombinant human ERbeta expressed in baculovirus expression system assessed as inhibition of estradiol-induced Eu...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Target4,4'-diapophytoene synthase(Staphylococcus aureus)
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of Staphylococcus aureus dehydrosqualene synthase expressed in Escherichia coli BL21 (DE3) cells by continuous spectrophotometric assayMore data for this Ligand-Target Pair
Target4,4'-diapophytoene synthase(Staphylococcus aureus)
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
University Of Illinois At Urbana-Champaign
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of Staphylococcus aureus dehydrosqualene synthase expressed in Escherichia coli BL21 (DE3) cells by continuous spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of FAM-LTERHKILHRLLQEGSPSD from ERbeta (unknown origin) (260 to 502 residues) expressed in Escherichia coli rosetta (DE3) after 1 hr by ...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Antagonist activity at full length recombinant human ERbeta expressed in baculovirus expression system assessed as inhibition of estradiol-induced Eu...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Antagonist activity at full length recombinant human ERbeta expressed in baculovirus expression system assessed as inhibition of estradiol-induced Eu...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of jack bean alpha-mannosidaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of jack bean alpha-mannosidaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of FAM-Bim peptide binding to human full-length N-terminal His6-tagged Bcl2 (2 to 206 residues) expressed in Escherichia coli S12 extract ...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 185nMAssay Description:Displacement of FAM-LTERHKILHRLLQEGSPSD from ERalpha (unknown origin) (302 to 552 residues) expressed in Escherichia coli rosetta (DE3) after 1 hr by...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of FAM-Bim peptide binding to human full-length N-terminal His6-tagged Bcl2 (2 to 206 residues) expressed in Escherichia coli S12 extract ...More data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase(Homo sapiens (Human))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Binding affinity to human GGPPSMore data for this Ligand-Target Pair
TargetGeranylgeranyl pyrophosphate synthase BTS1(Saccharomyces cerevisiae (Yeast))
Institute Of Biological Chemistry
Curated by ChEMBL
Institute Of Biological Chemistry
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Binding affinity to Saccharomyces cerevisiae GGPPSMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibition of FAM-Bim peptide binding to MCl1 (unknown origin) measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2-ABD expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of ROCK (unknown origin)More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:Inhibition of FAM-Bim peptide binding to MCl1 (unknown origin) measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Peking University Shenzhen Graduate School
Curated by ChEMBL
Peking University Shenzhen Graduate School
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:Antagonist activity at full length recombinant human ERbeta expressed in baculovirus expression system assessed as inhibition of estradiol-induced Eu...More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of FAM-Bim peptide binding to MCl1 (unknown origin) measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibition of FAM-Bim peptide binding to Bcl-xl (unknown origin) measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University Of Technology
Curated by ChEMBL
Dalian University Of Technology
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Inhibition of FAM-Bim peptide binding to MCl1 (unknown origin) measured after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranesMore data for this Ligand-Target Pair