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Found 155 with Last Name = 'zagotto' and Initial = 'g'
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11315(1,4-diamino-5,8-dihydroxy-9,10-dihydroanthracene-9...)
Affinity DataKi:  350nM ΔG°:  -36.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11313(1,8-dihydroxy-4-nitro-anthraquinone | 4,5-dihydrox...)
Affinity DataKi:  780nM ΔG°:  -34.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11314(1,8-dihydroxy-4-nitro-9H-xanthen-9-one | 1,8-dihyd...)
Affinity DataKi:  800nM ΔG°:  -34.4kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
Affinity DataKi:  1.85E+3nM ΔG°:  -32.4kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11316(1,8-dihydroxy-9,10-dihydroanthracene-9,10-dione | ...)
Affinity DataKi: >4.00E+4nM ΔG°: >-24.8kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Zea mays (Maize))
University of Padova

LigandPNGBDBM11317(1,8-dihydroxy-9H-xanthen-9-one | Xanthenone-relate...)
Affinity DataKi: >4.00E+4nM ΔG°: >-24.8kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181856(4-methyl-7-(2-oxocyclopentyloxy)-2H-chromen-2-one ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564382(CHEMBL4795023)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564384(CHEMBL4784643)
Affinity DataIC50:  320nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564388(CHEMBL4776391)
Affinity DataIC50:  330nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  330nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564381(CHEMBL4778120)
Affinity DataIC50:  360nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564387(CHEMBL4789806)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564385(CHEMBL4798710)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50252622(CHEMBL4070389)
Affinity DataIC50:  370nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  660nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564383(CHEMBL4783065)
Affinity DataIC50:  710nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564380(CHEMBL4799521)
Affinity DataIC50:  880nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564386(CHEMBL4796675)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564379(CHEMBL4792639)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of recombinant human CK2alpha (1 to 336 residues) expressed in Escherichia coli BL21 (DE3) using RRADDSDDDD as substrate incubated for 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSRSF protein kinase 1(Homo sapiens (Human))
University Of Trento

Curated by ChEMBL
LigandPNGBDBM50564378(CHEMBL4787157)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant human SRPK1 expressed in Escherichia coli using RS peptide as substrate incubated for 15 mins in presence of ATP by Kinase-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181854(9-(3-aminopropoxy)-7H-furo[3,2-g]chromen-7-one | C...)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of rat spleen LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of HIPK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha/beta/gamma(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of PKAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of DYRK1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of rat spleen SYKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50340957(8-nitro-2-(2,3,4-trihydroxyphenyl)naphthalene-1,4-...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50340956(5,8-dihydroxy-2-(2,3,4-trihydroxyphenyl)naphthalen...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181853(7-acetonyloxy-3-acetylamino-8-methoxycoumarin | CH...)
Affinity DataIC50:  6.43E+3nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181850(4-methyl-2H-benzofuro[3,2-g]chromen-2-one | CHEMBL...)
Affinity DataIC50:  7.24E+3nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of human recombinant GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Rattus norvegicus)
Università

Curated by ChEMBL
LigandPNGBDBM4078(6,7,13,14-tetrahydroxy-2,9-dioxatetracyclo[6.6.2.0...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of rat spleen FGRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181858(8-methoxy-4-methyl-7-(2-oxocyclohexyloxy)-2H-chrom...)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181851(5-methyl-2,3-dihydro-1H-8,10-dioxa-pentaleno[1,2-b...)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50340955(2-(2,4-dihydroxyphenyl)-8-hydroxy-1,4-naphthoquino...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181852(3-aminoacetamido-4'-methylfuro[3,2-g]coumarin | CH...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50340955(2-(2,4-dihydroxyphenyl)-8-hydroxy-1,4-naphthoquino...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of DYRK1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50340956(5,8-dihydroxy-2-(2,3,4-trihydroxyphenyl)naphthalen...)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of DYRK1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181857(5-methoxy-4-methyl-7-(2-oxocyclohexyloxy)-2H-chrom...)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50181861(3-amino-8-methoxy-4'-methylfuro[3,2-g]coumarin | C...)
Affinity DataIC50:  2.17E+4nMAssay Description:Inhibition of MAO-A activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of FgrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.47E+4nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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