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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
248
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.30nM
Assay Description:
Inhibition of human recombinant soluble MAO-B expressed in Pichia pastoris incubated for 30 mins prior to substrate addition measured after 60 mins b...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 3.90nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in Pichia pastoris incubated for 30 mins prior to substrate addition measured after 60 min...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 55nM
Assay Description:
Irreversible inhibition of recombinant human MAO-B expressed in baculovirus infected BT1 cells using benzylamine as substrate at 200 uM preincubated ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 90nM
Assay Description:
Competitive reversible inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 91nM
Assay Description:
Inhibition of human MAO-B expressed in BTI insect cells using p-tyramine as substrate after 60 mins
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 160nM
Assay Description:
The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 350nM
pH: 7.4
Assay Description:
Study medium contained 0.1 mL of sodium phosphate buffer (0.05 M, pH 7.4), various concentrations of the newly synthesized compounds or reference com...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 380nM
Assay Description:
Inhibition of recombinant human MAO-B using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...
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Target
Amine oxidase [flavin-containing] B
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 970nM
Assay Description:
Inhibition of bovine brain MAOB using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 970nM
Assay Description:
Reversible inhibition of recombinant human MAOB expressed in Pichia pastoris using varying levels of kynuramine as substrate measured after 5 mins by...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 970nM
Assay Description:
Reversible inhibition of MAO-B in Wistar rat assessed as inhibition constant followed by using clorgyline as substrate
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Amine oxidase [flavin-containing] B
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 970nM
Assay Description:
MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...
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Target
Amine oxidase [flavin-containing] B
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 970nM
Assay Description:
Inhibition of bovine brain mitochondrial MAO-B by fluorometric assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 970nM
Assay Description:
Inhibitory concentration for human Monoamine oxidase B
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 970nM
Assay Description:
Inhibition constant against human recombinant Monoamine oxidase-B
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Target
Amine oxidase [flavin-containing] B
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 970nM
Assay Description:
Inhibitory activity against monoamine oxidase B in isolated bovine brain mitochondria
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Target
Cytochrome P450 2B1
(Rattus norvegicus)
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.05E+3nM
Assay Description:
Mechanism based inhibition of rat cytochrome P450 CYP2B1 measured by 7-EFC O-deethylation activity
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 1.35E+3nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate by spectrophotometry-based Holt method
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 1.35E+3nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate after 60 mins by Lineweaver-Burk plot
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 1.35E+3nM
Assay Description:
Competitive inhibition of rat liver MAO-B after 60 mins using p-tyramine as substrate by spectrophotometry
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.35E+3nM
Assay Description:
Competitive inhibition of MAOB in rat liver homogenate by spectrophotometrically
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 1.93E+3nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
Ki: 1.96E+3nM
Assay Description:
Competitive inhibition of human recombinant MAO-B after 60 mins using p-tyramine as substrate by spectrophotometry
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Amine oxidase [flavin-containing] A
(Bos taurus)
Sapienza University of Rome
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.80E+3nM ΔG°: -32.3kJ/mole
pH: 7.4 T: 2°C
Assay Description:
MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...
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Amine oxidase [flavin-containing] A
(Bos taurus)
Sapienza University of Rome
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.80E+3nM
Assay Description:
Inhibition of bovine brain mitochondrial MAO-A by fluorometric assay
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Amine oxidase [flavin-containing] A
(Bos taurus)
Sapienza University of Rome
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.80E+3nM
Assay Description:
Inhibition of bovine brain MAOA using kinuramine as substrate preincubated for 30 mins prior to substrate addition measured after 30 mins by fluorome...
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5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 5.64E+3nM
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 5.68E+3nM
Assay Description:
Irreversible inhibition of recombinant human MAOB expressed in Pichia pastoris using varying levels of kynuramine as substrate measured after 5 mins ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 5.70E+3nM
Assay Description:
The activities of recombinant hMAO-A and hMAO-B were determined using p-tyramine as common substrate and calculated as 0.18 +/- 0.01 nmol/mg/min (n =...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 8.15E+3nM
pH: 7.4
Assay Description:
Study medium contained 0.1 mL of sodium phosphate buffer (0.05 M, pH 7.4), various concentrations of the newly synthesized compounds or reference com...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 9.06E+3nM
Assay Description:
Inhibition of human MAO-A expressed in BTI insect cells using p-tyramine as substrate after 60 mins
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 9.06E+3nM
Assay Description:
Competitive reversible inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 insect cells using p-tyramine as substrate assesse...
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D(2) dopamine receptor
(Homo sapiens (Human))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: >1.00E+4nM
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5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sri International
Curated by
PDSP K
i
Database
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: >1.00E+4nM
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.06E+4nM
Assay Description:
Competitive inhibition of rat liver MAO-A after 60 mins using p-tyramine as substrate by spectrophotometry
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.57E+4nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate after 60 mins by Lineweaver-Burk plot
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.69E+4nM
Assay Description:
Inhibition of recombinant human MAO-A using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additi...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 2.81E+4nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate incubated for 30 mins by Ample...
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Amine oxidase [flavin-containing] A
(Bos taurus)
Sapienza University of Rome
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.80E+4nM
Assay Description:
Inhibitory activity against monoamine oxidase A in isolated bovine brain mitochondria
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 3.80E+4nM
Assay Description:
Inhibtory concentration for rat Monoamine oxidase A
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 6.73E+4nM
Assay Description:
Competitive inhibition of human recombinant MAO-A after 60 mins using p-tyramine as substrate by spectrophotometry
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.06E+5nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate by spectrophotometry-based Holt method
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Ki: 1.06E+5nM
Assay Description:
Competitive inhibition of MAOA in rat liver homogenate by spectrophotometrically
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 0.0170nM
Assay Description:
Inhibition of human monoamine oxidase B
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.30nM
Assay Description:
Inhibition of human recombinant MAO-B using benzylamine hydrochloride as substrate assessed as H2O2 synthesis after 1 hr by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.30nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells by Amplex Red assay
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.80nM
Assay Description:
In vitro ability of the compound to inhibit Monoamine oxidase B activity in rat whole brain in vitro
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 3nM
Assay Description:
Inhibition of rat brain synaptosome MAO-B
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 3.60nM
Assay Description:
Inhibition of rat brain MAO-B using [14C]-phenylethylamine substrate after 20 mins
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 3.90nM
Assay Description:
Inhibition of rat brain synaptosome MAO-A
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 3.90nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected insect cell membranes using kynuramine as substrate preincubated for 30 mins followed by ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 5.5nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate preincubated for 15 m...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 5.5nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.10nM
Assay Description:
Inhibition of Sprague-Dawley rat liver MAO-B using p-tyramine as substrate preincubated for 15 mins and measured after 45 mins by resorufin-based flu...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.10nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus-infected insect cells using p-tyramine as substrate incubated for 30 mins prior to sub...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.10nM
Assay Description:
Inhibition of human MAO-B
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.60nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrate
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.70nM
Assay Description:
Inhibition of MAO-B in mitochondria-enriched Sprague-Dawley rat liver fractions using p-tyramine as substrate incubated for 30 mins prior to substrat...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.70nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate using [14C]-phenylethylamine as substrate preincubated for 30 mins followed by substrate addition measure...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.80nM
Assay Description:
Irreversible inhibition of human MAOB
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.80nM
Assay Description:
Inhibition of human brain MAO-B using [14C]-phenylethylamine substrate after 20 mins
More data for this Ligand-Target Pair
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of human MAO-B
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells using benzylamine as substrate preincubated for 1 h...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 7nM
Assay Description:
Irreversible inhibition of human cerebral cortex MAO-B using [14C]-phenylethylamin as substrate pretreated for 60 mins followed by substrate addition...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of MAOB
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 7nM
Assay Description:
Compound was evaluated for the time-dependence inhibition of MAO-B at 60 minutes preincubation periods
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 7.08nM
Assay Description:
Displacement of [3H]-Ro 16-6491 from MAO-B receptor in rat cerebral cortex
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 8nM
Assay Description:
Inhibition of [3H]U-69593 binding to recombinant human Opioid receptor kappa 1
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 8nM
Assay Description:
In vitro inhibitory activity on rat brain MAO-B.
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 9nM
Assay Description:
Inhibition of recombinant human MAOB using benzylamine as substrate after 30 mins by Amplex red based spectrophotometric analysis
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 9.40nM
Assay Description:
Compound was evaluated for the time-dependence inhibition of MAO-B at 30 minutes pre-incubation periods
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 9.90nM
Assay Description:
Compound was evaluated for the time-dependence inhibition of MAO-B at 20 minutes pre-incubation periods
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 10nM
Assay Description:
Inhibition of rat recombinant MAO-B expressed in baculovirus-infected insect cells using p-tyraimne substrate
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: <10nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 20 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 11nM
Assay Description:
Inhibition of recombinant human MAO-B using benzylamine as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins b...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 12nM
Assay Description:
Inhibition of recombinant human microsomal MAOB expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 15 ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 13nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in insect cells using kynuramine as substrate assessed as formation of 4-hydroxyquinoline measured ev...
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Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 13nM
Assay Description:
In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 13nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells assessed as kynuramine hydrobromide oxidation after 20 mins by spectrophotometric ana...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 13.9nM
Assay Description:
Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assay
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 15nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAO-B assessed as inhibition of production of hydrogen peroxide after 15 mins by the Amplex Red fluorimetric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells after 15 mins by fluorimetric assay
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human MAO-B assessed as inhibition of p-tyramine oxidation to p-hydroxyphenyl-acetaldehyde after 15 mins by fluorimetric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus-infected BTI insect cells assessed as using transformed p-tyramine after 15 mins by flu...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAOB using p-tyramine as substrate incubated for 15 mins by fluorimetric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decrease in H2O2...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 17nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using p-tyramine as substrate pretreated for 15 mins followe...
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 18nM
Assay Description:
Inhibition of MAO-A in rat whole brain homogenate in presence of selegiline
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 18nM
Assay Description:
Inhibition of human recombinant MAO-B preincubated for 30 mins followed by p-tyramine hydrochloride addition measured after 30 mins by Amplex red flu...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 18nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells preincubated for 15 mins
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 18.5nM
Assay Description:
Inhibition of human recombinant MAOB assessed as H2O2 production by Amplex Red reagent-based assay
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 19nM
Assay Description:
Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells by para-tyramine oxidation assay
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as inhibition of hydrogen peroxide product...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19nM
Assay Description:
Inhibition of human recombinant MAO-B using benzylamine as substrate incubated for 15 mins prior to substrate addition measured after 20 mins by fluo...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate incubated for 15 mins prior to substrate...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAO-B using p-tyramine substrate by flurometric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramin...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAOB expressed in BTI insect cells using p-tyramine substrate by fluorometric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAOB
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAOB by fluorimetric method
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI-TN-5B1-4 insect sells assessed as hydrogen peroxide production by fluorim...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 19.6nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BT1-TN-5B1-4 cells assessed as inhibition of production of hydrogen peroxide ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus-infected insect BTI-TN-5B1-4 cells assessed as p-tyramine conversion to H2O...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as reduc...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 production
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate using [14C]-5HT as substrate preincubated for 30 mins followed by substrate addition measured after 20 mi...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus-infected BTI-TN-5B1-4 cell microsomes assessed as decrease in H2O2 production using p-...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in baculovirus infected BT1 cells
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 20nM
pH: 7.4 T: 2°C
Assay Description:
The effects of the test compounds on hMAO isoform enzymatic activity were evaluated by measuring their effects on the production of hydrogen peroxide...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human MAO-B assessed as inhibition of H2O2 production using p-tyramine as substrate
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected insect BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-t...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as produ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 20 mins by fluorescence assay
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAOB expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human recombinant MAOB using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 20nM
Assay Description:
Inhibition of human MAO-B using p-tyramine as substrate after 15 mins by amplex red reagent based assay
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Target
Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 25nM
Assay Description:
Inhibitory activity against rat brain mitochondrial Monoamine oxidase
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 33nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells using p-tyramine as substrate preincubated for 30 mins followed by substrate addition...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 36nM
Assay Description:
Inhibition of MAO-B (unknown origin)
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 39nM
Assay Description:
Inhibition of human microsomal MAO-B expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in 4-hydroxyquinoline formation using...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 40nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using tyramine as substrate pretreated for 30 mins followed ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 40nM
Assay Description:
Inhibition of human MAO-B using tyramine hydrochloride as substrate preincubated for 30 mins followed by substrate addition and measured after 30 min...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 42nM
Assay Description:
Inhibition of human MAO-B expressed in baculovirus infected insect cell membranes using kynuramine as substrate after 15 to 20 mins by discontinuous ...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 43nM
Assay Description:
Inhibition of MAO-B (unknown origin) by fluorometric assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 44nM
Assay Description:
Inhibition of human MAO-B using tyramine hydrochloride as substrate after 30 mins by Amplex Red reagent based horseradish peroxidase enzyme-coupled f...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 45nM
Assay Description:
Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 52nM
Assay Description:
Inhibition of Monoamine oxidase B of rat liver mitochondrial membranes
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 56nM
Assay Description:
Inhibition of recombinant human MAO-B assessed as inhibition of kynuramine oxidation by spectrophotometry
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 60nM
Assay Description:
Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 30 mins follow...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 67.3nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramin...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 70nM
Assay Description:
Inhibition of MAO-B (unknown origin)
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 71nM
Assay Description:
Inhibition of MAO-B (unknown origin) using (4S)-4,5-dihydro-2-(6-hydroxybenzothiazolyl)-4-thiazolecarboxylic acid as substrate by MAO-Glo assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of MAO-B (unknown origin)
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of human recombinant monoamine oxidase-B assessed as kynuramine conversion to 6-hydroxyquinoline after 20 mins by fluorescence spectrophot...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells microsomes assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate after 20 mins by fluorescence spectrophotometric analysis
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of human recombinant MAOB expressed in insect cell microsomes using kynuramine as substrate after 20 mins by fluorescence spectrophotometr...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 79nM
Assay Description:
Inhibition of recombinant human MAO-B using kynuramine as substrate by fluorescence spectroscopy
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 85.2nM
Assay Description:
Inhibition of human recombinant MAO-B expressed in insect cells assessed as inhibition of kynuramine oxidation after 30 mins by fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 94nM
Assay Description:
Inhibition of MAOB (unknown origin) using beetle luciferin as substrate by MAO-Glo assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 95nM
Assay Description:
Inhibition of human recombinant MAOB using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometry
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Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 160nM
Assay Description:
Compound was evaluated for the time-dependence inhibition of MAO-B at 0 minute pre-incubation periods
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 221nM
Assay Description:
Inhibition of recombinant human MAO-B expressed in Sf9 cells using benzylamine as substrate preincubated for 15 mins followed by substrate addition f...
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Alpha-synuclein
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: 270nM
Assay Description:
Inhibition of alpha-synuclein fibril formation (unknown origin) incubated for 6 days by thioflavin S based fluorescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 270nM
Assay Description:
Inhibition of human recombinant MAOB
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Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 280nM
Assay Description:
Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 M
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 321nM
Assay Description:
Inhibition of recombinant human microsomal MAO-B expressed in baculovirus-infected insect cells using p-tyramine as substrate assessed as H2O2 produc...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 334nM
Assay Description:
Inhibition of human MAOB after 1 hr by luminescence assay
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 480nM
Assay Description:
Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 516nM
Assay Description:
In vitro ability of the compound to inhibit Monoamine oxidase A activity in rat whole brain in vitro
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Target
Amine oxidase [flavin-containing] A/B
(Rattus norvegicus (rat))
TBA
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 650nM
Assay Description:
In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 700nM
Assay Description:
Compound was evaluated for the time-dependence inhibition of MAO-A at 60 minutes of preincubated period. values are same with or without pre-incubati...
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 800nM
Assay Description:
In vitro inhibitory activity on rat brain by monoamine oxidase A (MAO-A)
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 944nM
Assay Description:
Inhibition of rat brain MAO-A using [14C]-5- hydroxytryptamine creatinine disulphate substrate after 30 mins
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 969nM
Assay Description:
Inhibition of Sprague-Dawley rat liver MAO-A using p-tyramine as substrate preincubated for 15 mins and measured after 45 mins by resorufin-based flu...
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Target
Amine oxidase [flavin-containing] B
(Bos taurus)
National Research Center
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of bovine mitochondrial MAOB
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.20E+3nM
Assay Description:
Inhibition of MAOA
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.20E+3nM
Assay Description:
Displacement of [3H]-Ro 41-1049 from MAO-A receptor in rat cerebral cortex
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.42E+3nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as decrease in H2O2 production using p-tyr...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.42E+3nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells using p-tyramine as substrate preincubated for 15 m...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.50E+3nM
Assay Description:
Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins by...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.60E+3nM
Assay Description:
Competitive inhibition of MAOB in rat liver homogenate by spectrophotometrically
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.70E+3nM
Assay Description:
Inhibition of human brain MAO-A using [14C]-5- hydroxytryptamine creatinine disulphate substrate after 30 mins
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.70E+3nM
Assay Description:
Irreversible inhibition of human cerebral cortex MAO-A using [14C]-5-hydroxytryptamine creatinine disulphate as substrate pretreated for 60 mins foll...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.86E+3nM
Assay Description:
Inhibition of rat mitochondrial MAO-B using DAB as substrate incubated for 30 mins by HPLC analysis
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.00E+3nM
Assay Description:
Inhibition of human recombinant MAO-A preincubated for 30 mins followed by p-tyramine hydrochloride addition measured after 30 mins by Amplex red flu...
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.01E+3nM
Assay Description:
Inhibition of MAOB in rat liver homogenates preincubated for 60 mins
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Target
Amine oxidase [flavin-containing] B
(Rattus norvegicus (rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.01E+3nM
Assay Description:
Inhibition of MAO-B in rat liver homogenate after 60 mins by residual activity plot
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.09E+3nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells using tyramine as substrate preincubated for 1 hr f...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.82E+3nM
Assay Description:
Inhibition of human recombinant MAO-B using p-tyramine as substrate assessed as production of H2O2 incubated for 15 mins prior to substrate addition ...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.89E+3nM
Assay Description:
Inhibition of recombinant human MAOB using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additio...
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 3.80E+3nM
Assay Description:
Inhibition of Monoamine oxidase A of rat liver mitochondrial membranes
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 9.70E+3nM
Assay Description:
A stock solution was prepared using a human MAO-B enzyme (purchased from Aldrich) and a Amplex Red monoamine oxidase assay kit according to a prepara...
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.10E+4nM
Assay Description:
Inhibition of MAO-B (unknown origin) using p-tyramine substrate by HPLC method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.91E+4nM
Assay Description:
Inhibitory activity of compounds was evaluated by a homogeneous luminescent method, the MAO-Glo Assay (Promega), measuring the monoamine oxidase acti...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.96E+4nM
Assay Description:
Inhibition of human MAOB by fluorimetry
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.96E+4nM
Assay Description:
Inhibition of human MAOB expressed in BTI insect cells
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 1.96E+4nM
Assay Description:
Inhibition of human recombinant MAOB
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.01E+4nM
Assay Description:
Inhibition of human microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells assessed as reduction in 4-hydroxyquinoline formation using...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 2.97E+4nM
Assay Description:
Inhibition of human recombinant MAOA using kynuramine substrate incubated for 20 mins by fluorescence spectrophotometry
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of human MAO-A expressed in baculovirus infected insect cell membranes using kynuramine as substrate after 15 to 20 mins by discontinuous ...
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Amine oxidase [flavin-containing] A
(Bos taurus)
Sapienza University of Rome
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: 3.80E+4nM
Assay Description:
Inhibition of bovine mitochondrial MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 4.79E+4nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 5.43E+4nM
Assay Description:
Inhibition of recombinant human MAOA expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 30 mins follow...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 5.44E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in insect cells using p-tyramine as substrate preincubated for 30 mins followed by substrate addition...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 5.54E+4nM
Assay Description:
Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: >6.00E+4nM
Assay Description:
Inhibition of recombinant human MAOA using p-tyramine as substrate assessed as H2O2 production preincubated for 15 mins followed by substrate additio...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.27E+4nM
Assay Description:
Inhibition of recombinant human microsomal MAOA expressed in baculovirus infected BTI insect cells using p-tyramine as substrate preincubated for 15 ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.28E+4nM
Assay Description:
Inhibition of human MAO-A assessed as inhibition of H2O2 production using p-tyramine as substrate
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.36E+4nM
Assay Description:
Inhibition of human MAO-A expressed in baculovirus infected BTI insect cells preincubated for 15 mins
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.72E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 production
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as hydrogen peroxide production from p-tyra...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate incubated for 15 mins prior to substrate...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Displacement of [3H]R-1881 from Androgen receptor of LNCaP cells
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of recombinant human MAO-A using kynuramine as substrate after 20 mins by fluorescence assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as produ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus-infected insect BTI-TN-5B1-4 cells assessed as p-tyramine conversion to H2O...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.73E+4nM
pH: 7.4 T: 2°C
Assay Description:
The effects of the test compounds on hMAO isoform enzymatic activity were evaluated by measuring their effects on the production of hydrogen peroxide...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus-infected BTI-TN-5B1-4 cell microsomes assessed as decrease in H2O2 production using p-...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAO-A expressed in baculovirus infected BTI-TN-5B1-4 cells using p-tyramine as substrate assessed as reduc...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in BTI cells
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells by para-tyramine oxidation assay
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human MAOA expressed in BTI insect cells
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human MAOA by fluorimetry
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus infected insect BTI-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-t...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect sells assessed as hydrogen peroxide production by fluorim...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in BTI-TN-5B1-4 cells assessed as H2O2 production using para-tyramine substrate by fluorimetric metho...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in BTI insect cells using p-tyramine substrate by fluorometric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A using p-tyramine substrate by flurometric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in insect BT1-TN-5B1-4 cells assessed as production of hydrogen peroxide from p-tyramine up to 15 min...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN-5B1-4 insect cells assessed as inhibition of hydrogen peroxide product...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.73E+4nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BT1-TN-5B1-4 cells assessed as inhibition of production of hydrogen peroxide ...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.76E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BT1 cells
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant MAOA using p-tyramine as substrate incubated for 15 mins by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using p-tyramine as substrate pretreated for 15 mins followe...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human MAO-A assessed as inhibition of p-tyramine oxidation to p-hydroxyphenyl-acetaldehyde after 15 mins by fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant MAOA expressed in baculovirus-infected BTI insect cells assessed as conversion of p-tyramine into p-hydroxyphenyl-ace...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI-TN5B1-4 cells using p-tyramine as substrate assessed as reduction in H2O2...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Copy SMILES
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 6.87E+4nM
Assay Description:
Inhibition of human recombinant MAO-A assessed as inhibition of production of hydrogen peroxide after 15 mins by Amplex Red fluorimetric method
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Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 7.02E+4nM
Assay Description:
Inhibition of human recombinant MAOA assessed as H2O2 production by Amplex Red reagent-based assay
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
Birla Institute of Technology
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 7.02E+4nM
Assay Description:
Inhibition of human recombinant MAO-A using p-tyramine as substrate incubated for 15 mins prior to substrate addition measured after 20 mins by fluor...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: 9.06E+4nM
Assay Description:
Competitive inhibition of MAOA in rat liver homogenate by spectrophotometrically
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Target
Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assay
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ATP-binding cassette sub-family C member 3
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...
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ATP-binding cassette sub-family C member 4
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
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ATP-binding cassette sub-family C member 2
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
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Bile salt export pump
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >1.33E+5nM
Assay Description:
Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...
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Target
Bile salt export pump
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >1.35E+5nM
Assay Description:
Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: 4.99E+5nM
Assay Description:
Inhibition of MAOA in rat liver homogenates preincubated for 60 mins
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Amine oxidase [flavin-containing] A
(Rattus norvegicus (rat))
Birla Institute Of Technology
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
IC50: 4.99E+5nM
Assay Description:
Inhibition of MAO-A in rat liver homogenate after 60 mins by residual activity plot
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Acetylcholinesterase
(Homo sapiens (Human))
Okayama University
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >5.00E+5nM
Assay Description:
Inhibition of human recombinant AChE expressed in HEK293 cells using acetylthiocholine iodide as substrate preincubated for 30 mins followed by subst...
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Cholinesterase
(Homo sapiens (Human))
Okayama University
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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IC50: >5.00E+5nM
Assay Description:
Inhibition of human recombinant BuChE expressed in HEK293 cells using S-butyrylthiocholine iodide as substrate preincubated for 30 mins followed by s...
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Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Dart Neuroscience
Curated by
ChEMBL
Ligand
BDBM15579
(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
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Affinity Data
Kd: 59nM
Assay Description:
Binding affinity to human recombinant microsomal MAO-B by ITC
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