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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
65
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 18nM
Assay Description:
Binding affinity to human adrenergic alpha1A receptor by radioligand displacement assay
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 40nM
Assay Description:
Binding affinity to human adrenergic Alpha-1D receptor by radioligand displacement assay
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 65nM
Assay Description:
Binding affinity to human adrenergic Alpha-1B receptor by radioligand displacement assay
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 77nM
Assay Description:
Binding affinity to human dopamine D2S receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: 280nM
Assay Description:
Binding affinity to human 5-HT1A receptor by radioligand displacement assay
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: 530nM
Assay Description:
Binding affinity to human adrenergic alpha2A receptor by radioligand displacement assay
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Target
Histamine H1 receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 610nM
Assay Description:
Binding affinity to human histamine H1 receptor by radioligand displacement assay
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Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 840nM
Assay Description:
Binding affinity to adrenergic alpha2B receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 891nM
Assay Description:
Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...
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Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 980nM
Assay Description:
Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...
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Target
Adenosine receptor A1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human adenosine A1 receptor by radioligand displacement assay
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Target
Melanocortin receptor 4
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human MC4 receptor by radioligand displacement assay
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Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT2A agonist site receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human muscarinic M1 receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT2B agonist site receptor by radioligand displacement assay
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Target
Histamine H3 receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human histamine H3 receptor by radioligand displacement assay
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Target
Mu-type opioid receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human mu opioid receptor agonist site by radioligand displacement assay
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human adrenergic beta-1 receptor by radioligand displacement assay
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Target
Gastrin/cholecystokinin type B receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human CCK2 receptor by radioligand displacement assay
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Target
Substance-P receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human NK1 receptor by radioligand displacement assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to adrenergic beta2 receptor by radioligand displacement assay
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Target
High affinity choline transporter 1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human choline transporter (CHT1) by radioligand displacement assay
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Target
Adenosine receptor A2a
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human adenosine A2A receptor by radioligand displacement assay
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Target
Ribosyldihydronicotinamide dehydrogenase [quinone]
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to ML2 (MT3) receptor by radioligand displacement assay
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Target
Cannabinoid receptor 1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human CB1 receptor by radioligand displacement assay
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Target
Kappa-type opioid receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to kappa opioid receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT7 receptor by radioligand displacement assay
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Target
Sodium-dependent noradrenaline transporter
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human NE transporter by radioligand displacement assay
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Target
Substance-K receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human NK2 receptor by radioligand displacement assay
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Target
Neurotensin receptor type 1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human UT1 receptor by radioligand displacement assay
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human D2S agonist site receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M4
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human muscarinic M4 receptor by radioligand displacement assay
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Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human dopamine transporter by radioligand displacement assay
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NCI pathway
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Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT4e receptor by radioligand displacement assay
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Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to p38alpha by radioligand displacement assay
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Target
Acetylcholinesterase
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human acetylcholine esterase by radioligand displacement assay
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human dopamine D3 receptor by radioligand displacement assay
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Target
Neuropeptide Y receptor type 1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human neuropeptide Y1 receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human muscarinic M2 receptor by radioligand displacement assay
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Target
Melatonin receptor type 1A
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human MT1 receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human muscarinic M3 receptor by radioligand displacement assay
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Target
Adenosine receptor A1
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human adenosine A1 receptor agonist site by radioligand displacement assay
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Target
Endothelin-1 receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human ETA receptor by radioligand displacement assay
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Target
Glucocorticoid receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human glucocorticoid receptor by radioligand displacement assay
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Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to Lyn by radioligand displacement assay
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human dopamine D1 receptor by radioligand displacement assay
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Target
Nischarin
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to I1 receptor by radioligand displacement assay
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Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to MAOA by radioligand displacement assay
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Target
Sodium-dependent serotonin transporter
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT transporter by radioligand displacement assay
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Target
Histamine H2 receptor
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human histamine H2 receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 2C
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5HT2C receptor agonist site by radioligand displacement assay
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Target
Neuronal acetylcholine receptor subunit alpha-4/beta-2
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to nAChR alpha4beta2 receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human 5-HT3 receptor by radioligand displacement assay
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to 5-HT1B receptor by radioligand displacement assay
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Target
Adenosine receptor A3
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Binding affinity to human adenosine A3 receptor by radioligand displacement assay
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Target
Muscarinic acetylcholine receptor M5
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: <1.00E+3nM
Assay Description:
Agonist activity at human muscarinic M5 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assay
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Target
Muscarinic acetylcholine receptor M4
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 1.40E+3nM
Assay Description:
Agonist activity at human muscarinic M4 receptor expressed in BHK-21 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 1.74E+3nM
Assay Description:
Displacement of [3H]NMS from EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 22 hrs by liquid scinti...
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Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 2.80E+3nM
Assay Description:
Agonist activity at human muscarinic M3 receptor expressed in BHK-21 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assay
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Target
Muscarinic acetylcholine receptor M5
(Homo sapiens (Human))
H. Lundbeck
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
Ki: 4.50E+3nM
Assay Description:
Displacement of [3H]-4-DAMP from human muscarinic M5 receptor expressed in BHK-21 cells
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
EC50: 150nM
Assay Description:
Agonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assay
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
EC50: 740nM
Assay Description:
Partial agonist activity at human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluorescence assay
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
EC50: 720nM
Assay Description:
Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 11 residues expressed in HEK293 cells assessed as induction of calci...
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
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Affinity Data
EC50: 450nM
Assay Description:
Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as induction of calci...
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
University Of Strasburg
Curated by
ChEMBL
Ligand
BDBM50326219
(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 210nM
Assay Description:
Partial agonist activity at EGFP-fused human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluoresce...
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