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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Histamine H3 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50321816
(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
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Affinity Data
Ki: 5.40nM
Assay Description:
Displacement of [3H] (R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Histamine H1 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50321816
(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Displacement of [3H]rilamine from human histamine H1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H2 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50321816
(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Displacement of [125I]aminopotentidine from human histamine H2 receptor expressed in CHO-K1 cells after 1 hr by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50321816
(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
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Affinity Data
Ki: 3.10E+3nM
Assay Description:
Displacement of [3H]histamine from human histamine H4 receptor expressed in CHO-K1 cells after 1 hr by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Meiji Seika Kaisha
Curated by
ChEMBL
Ligand
BDBM50321816
(4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)pi...)
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Copy InChI
Affinity Data
EC50: 7.60nM
Assay Description:
Agonist activity at human recombinant histamine H3 receptor expressed in CHO-K1 cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintil...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI