Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 45 hits in this display
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 1.71E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 2.80E+4nMAssay Description:Inhibition of PRL-3-mediated cell migration in human DLD1 cells after 15 hrs by crystal violet staining based microscopic assayMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 3.20E+4nMAssay Description:Inhibition of bovine kidney alpha-fucosidase using PNPG as substrate incubated for 10 mins by spectrophotometric methodMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 3.50E+4nMAssay Description:Inhibition of PRL-3-mediated cell invasion in human DLD1 cells after 20 hrs using crystal violet staining by Matrigel invasion assayMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 4.31E+4nMpH: 7.0 T: 2°CAssay Description:The enzymatic activities of FtFabZ and YpFabZ were determined via the reportedspectrophotometric method using the substrate analogue crotonoyl-CoA.7 ...More data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 5.20E+4nMAssay Description:Compound was tested for the enzyme inhibitory activity against Human Leukocyte Elastase (HLE) at 53 uM concentrationMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 1.25E+5nMAssay Description:SDFQ HTS primary assay using pAB1_FL905 was performed in 2 µL of (1 xDNA gyrase buffer: 20 mM Tris-Acetate pH 7.9, 50 mM KAc, 10 mM MgCl2, 2 mM DTT, ...More data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)
IC50: 7.60E+5nMAssay Description:Inhibition of human Neu2 assessed as MuNANA substrate hydrolysis in presence of 0.1% Triton X-100 by discontinuous fluorimetric assayMore data for this Ligand-Target Pair
BDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)