Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM410099(US10370370, Compound 3-P1)
BDBM410101(US10370370, Compound (R)-3)
Ki: 57nMAssay Description:h-5HT3: In brief, Chinese Hamster Ovary (CHO) cells stably expressing human 5-HT3 serotonin receptors, grown to confluence in 175 cm2 flasks. Followi...More data for this Ligand-Target Pair
BDBM410100(US10370370, Compound 3-P2)
BDBM410100(US10370370, Compound 3-P2)
Ki: 458nMAssay Description:h-5HT3: In brief, Chinese Hamster Ovary (CHO) cells stably expressing human 5-HT3 serotonin receptors, grown to confluence in 175 cm2 flasks. Followi...More data for this Ligand-Target Pair
BDBM410099(US10370370, Compound 3-P1)
Ki: 1.40E+3nMAssay Description:α7 nAChR: The ability of compounds to displace binding of radioactive ligands from human α7 nAChR was determined, as a measure of the affin...More data for this Ligand-Target Pair