Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 47 hits in this display
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
Arginase(Leishmania amazonensis)Universidade Federal De S£O Carlos
Curated by ChEMBL
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
Ki: 5.60E+3nMpH: 7.4Assay Description:Carbonic anhydrase activity was assayed by following the change in absorbance at 348 nm of 4-nitrophenylacetate (NPA) to 4-nitrophenylate ion over a ...More data for this Ligand-Target Pair
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
Ki: 6.80E+3nMpH: 7.4Assay Description:Carbonic anhydrase activity was assayed by following the change in absorbance at 348 nm of 4-nitrophenylacetate (NPA) to 4-nitrophenylate ion over a ...More data for this Ligand-Target Pair
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
Arginase(Leishmania amazonensis)Universidade Federal De S£O Carlos
Curated by ChEMBL
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
IC50: 2.02E+4nMAssay Description:Inhibition of cyclooxygenase activity of COX1 in sheep seminal vesicle in presence of 1 mM phenol by cyclooxygenase assayMore data for this Ligand-Target Pair
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
IC50: 2.41E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
IC50: 1.00E+5nMAssay Description:Inhibition of recombinant oligo-histidine-tagged Leishmania major DHODH expressed in Escherichia coli BL21(DE3) cells using DHO as substrate measured...More data for this Ligand-Target Pair
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
IC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute(SBMRI, San Diego, CA...More data for this Ligand-Target Pair
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
IC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
BDBM60836((+)-Catechin hydrate | (2R,3S)-2-(3,4-dihydroxyphe...)
IC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
EC50: 4.73E+4nMAssay Description:Agonist activity at human MT2R stably expressed in HEK293 cells by FlexStation3 Bench-top MultiMode Microplate ReaderMore data for this Ligand-Target Pair
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
BDBM23416(α-CA inhibitor, 3 | (+)-Catechin | (2R,3S)-2-...)
EC50: 2.58E+4nMAssay Description:Agonist activity at human MT1R stably expressed in HEK293 cells by FlexStation3 Bench-top MultiMode Microplate ReaderMore data for this Ligand-Target Pair