Compile Data Set for Download or QSAR
maximum 50k data
Found 389 Enz. Inhib. hit(s) with all data for entry = 50001811
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397215(CHEMBL2172295)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397206(CHEMBL2172289)
Affinity DataKi:  5.69nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50370108(CHEMBL1790713)
Affinity DataKi:  6.24nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307120(5-[4-[(1,1'-Biphenyl-2-ylcarbonyl)amino]-3-methylb...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50370109(CHEMBL1790723)
Affinity DataKi:  7.60nMAssay Description:Binding affinity for human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397213(CHEMBL2172391)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM212437(JMV 3011)
Affinity DataKi:  8.30nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  8.70nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397219(CHEMBL2172285)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1 [E24Q](Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataKi:  8.90nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397210(CHEMBL2172290)
Affinity DataKi:  9.02nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  9.20nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.70nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Growth hormone secretagogue receptor type 1(Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  9.90nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataKi:  9.90nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50459392(CHEMBL4216873)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459394(CHEMBL4215258)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459394(CHEMBL4215258)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459396(CHEMBL4209266)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459401(CHEMBL4210854)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50459394(CHEMBL4215258)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459410(CHEMBL4209421)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459413(CHEMBL4218739)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50094081((4-Amino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepi...)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459412(CHEMBL4207413)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50459407(CHEMBL4204008)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50459396(CHEMBL4209266)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459396(CHEMBL4209266)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50459392(CHEMBL4216873)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50459395(CHEMBL4210158)
Affinity DataKi: <10nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Growth hormone secretagogue receptor type 1(Homo sapiens (Human))
Université Montpellier 1

LigandPNGBDBM50049478(1-{[(2R)-3-(benzyloxy)-1-{1-methanesulfonyl-1,2-di...)
Affinity DataKi:  10.2nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50370113(CHEMBL1790719)
Affinity DataKi:  11.8nMAssay Description:Binding affinity for human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50370117(CHEMBL1790720)
Affinity DataKi:  12.2nMAssay Description:Binding affinity for human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397212(CHEMBL2172392)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50139178(CHEMBL3763342)
Affinity DataKi:  13nMAssay Description:Displacement of DY647 from SNAP-tagged V1A receptor (unknown origin) expressed in HEK293 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50370115(CHEMBL1790717)
Affinity DataKi:  13.7nMAssay Description:Binding affinity for human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397216(CHEMBL2172294)
Affinity DataKi:  14.1nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  14.1nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397209(CHEMBL2172291)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50397211(CHEMBL2172393)
Affinity DataKi:  16.8nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50307118(5-[2-Chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-1...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-AVP from human OXR receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50307118(5-[2-Chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-1...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]AVP from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50370112(CHEMBL1790729)
Affinity DataKi:  17.3nMAssay Description:Binding affinity for human Vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50103476(CHEMBL412559 | Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50307119(1-Methyl-5-[3-methyl-4-(3-methyl-1H-pyrazol-1-yl)b...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Institute Genomics Functional (Igf)

Curated by ChEMBL
LigandPNGBDBM50166223(CHEMBL265137 | Vasopressin Analogue)
Affinity DataKi:  18nMAssay Description:Binding affinity against human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM212436(JMV 3002 | N-[1-[4-[(2,4-dimethoxyphenyl)methyl]-5...)
Affinity DataKi:  19.3nMAssay Description:Briefly, direct ligand binding experiments were performed using fluorescence energy transfer with the purified receptor labeled with Alexa Fluor 350 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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