Compile Data Set for Download or QSAR
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Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 3112
LigandPNGBDBM28194(3-[(3-chlorothiophen-2-yl)methoxy]-5-(5,6-dimethox...)
Affinity DataIC50:  2nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28200(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(t...)
Affinity DataIC50:  2nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28175(5-(6-methoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(trifl...)
Affinity DataIC50:  2nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25120(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(t...)
Affinity DataIC50:  2nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28177(3-[(2-bromophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3...)
Affinity DataIC50:  2nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28178(3-[(2-chlorophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,...)
Affinity DataIC50:  2nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28169(5-(6-chloro-1H-1,3-benzodiazol-1-yl)-3-[(2-methylp...)
Affinity DataIC50:  4nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28182(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(t...)
Affinity DataIC50:  5nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28179(3-[(2-cyanophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3...)
Affinity DataIC50:  6nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28202(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(t...)
Affinity DataIC50:  6nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28174(5-(5-methoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(trifl...)
Affinity DataIC50:  8nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28183(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-[(2-me...)
Affinity DataIC50:  8nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25120(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2-(t...)
Affinity DataIC50:  9nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28171(3-[(2-bromophenyl)methoxy]-5-[6-(trifluoromethyl)-...)
Affinity DataIC50:  9nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28192(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(thiop...)
Affinity DataIC50:  11nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28166(5-(1H-1,3-benzodiazol-1-yl)-3-[(2-bromophenyl)meth...)
Affinity DataIC50:  11nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28173(5-(6-methanesulfonyl-1H-1,3-benzodiazol-1-yl)-3-{[...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28162(5-(1H-1,3-benzodiazol-1-yl)-3-[(2-chlorophenyl)met...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28159(5-(1H-1,3-benzodiazol-1-yl)-3-[(2-methoxyphenyl)me...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28158(5-(1H-1,3-benzodiazol-1-yl)-3-[(3-methylphenyl)met...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28157(5-(1H-1,3-benzodiazol-1-yl)-3-[(2-methylphenyl)met...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28176(3-(benzyloxy)-5-(5,6-dimethoxy-1H-1,3-benzodiazol-...)
Affinity DataIC50:  12nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28187(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-[(4-me...)
Affinity DataIC50:  13nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28167(5-(1H-1,3-benzodiazol-1-yl)-3-[(2-fluorophenyl)met...)
Affinity DataIC50:  14nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28198(3-[(2-bromopyridin-4-yl)methoxy]-5-(5,6-dimethoxy-...)
Affinity DataIC50:  14nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28165(5-(1H-1,3-benzodiazol-1-yl)-3-{[2-(trifluoromethyl...)
Affinity DataIC50:  15nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28193(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(thiop...)
Affinity DataIC50:  17nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28181(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-[(2-ac...)
Affinity DataIC50:  17nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28191(3-(cyclohexylmethoxy)-5-(5,6-dimethoxy-1H-1,3-benz...)
Affinity DataIC50:  17nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28185(3-[(3-aminophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3...)
Affinity DataIC50:  21nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28168(5-(5-chloro-1H-1,3-benzodiazol-1-yl)-3-[(2-methylp...)
Affinity DataIC50:  21nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28163(5-(1H-1,3-benzodiazol-1-yl)-3-[(3-chlorophenyl)met...)
Affinity DataIC50:  22nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28195(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(furan...)
Affinity DataIC50:  27nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28160(5-(1H-1,3-benzodiazol-1-yl)-3-[(3-methoxyphenyl)me...)
Affinity DataIC50:  28nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28184(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[3-(d...)
Affinity DataIC50:  31nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28180(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-[(2-me...)
Affinity DataIC50:  31nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28190(3-(cyclopentylmethoxy)-5-(5,6-dimethoxy-1H-1,3-ben...)
Affinity DataIC50:  34nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28161(5-(1H-1,3-benzodiazol-1-yl)-3-[(4-methoxyphenyl)me...)
Affinity DataIC50:  35nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28189(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(3-phe...)
Affinity DataIC50:  61nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28156(5-(1H-1,3-benzodiazol-1-yl)-3-(benzyloxy)thiophene...)
Affinity DataIC50:  61nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27443(5-(1H-1,3-benzodiazol-1-yl)-3-[(4-methylphenyl)met...)
Affinity DataIC50:  70nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28201(5,6-dimethoxy-1-[5-(1H-1,2,3,4-tetrazol-5-yl)-4-{[...)
Affinity DataIC50:  73nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27444(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-[(4-me...)
Affinity DataIC50:  75nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28203(1-[5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-{[2...)
Affinity DataIC50:  85nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28186(3-[(3-cyanophenyl)methoxy]-5-(5,6-dimethoxy-1H-1,3...)
Affinity DataIC50:  99nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28164(5-(1H-1,3-benzodiazol-1-yl)-3-[(4-chlorophenyl)met...)
Affinity DataIC50:  100nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28188(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(2-phe...)
Affinity DataIC50:  130nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28197(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(pyrid...)
Affinity DataIC50:  130nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28196(5-(5,6-dimethoxy-1H-1,3-benzodiazol-1-yl)-3-(furan...)
Affinity DataIC50:  190nMAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28172(5-(5-methanesulfonyl-1H-1,3-benzodiazol-1-yl)-3-{[...)
Affinity DataIC50:  250nMpH: 7.2 T: 22°CAssay Description:The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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