Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50033491
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.416nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 387nMAssay Description:Displacement of [3H]SP from human recombinant NK1 receptor expressed in CHO cells after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 445nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes after 2 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
Affinity DataIC50: 8.51nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 43.3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
Affinity DataKd: 31.6nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 631nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 3.98nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair
Affinity DataKd: 15.8nMAssay Description:Antagonist activity at human NK1 receptor expressed in CHO-K1 cells assessed as inhibition of substance P-induced calcium-dependent aequorine lumines...More data for this Ligand-Target Pair