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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM135630'
TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM135630(US10179804, Example 15 | US10632171, Peptide No. 1...)
Affinity DataKi:  0.700nMpH: 7.5Assay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM135630(US10179804, Example 15 | US10632171, Peptide No. 1...)
Affinity DataKi:  0.700nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM135630(US10179804, Example 15 | US10632171, Peptide No. 1...)
Affinity DataKi:  0.700nMAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM135630(US10179804, Example 15 | US10632171, Peptide No. 1...)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/moleT: 37°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In DepthDetails US Patent