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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50045488'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50045488(CHEMBL3310123)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]Mesulergine from human 5-HT2B receptor expressed in HEK293-EBNA cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50045488(CHEMBL3310123)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50045488(CHEMBL3310123)
Affinity DataIC50:  52nMAssay Description:Inhibition of human 5-HT2B receptor expressed in HEK293-EBNA cells assessed as [3H]PI metabolism by by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed