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Found 2 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM10520'
TargetAcetylcholinesterase(Homo sapiens (Human))
Universita Degli Studi Di Siena

LigandPNGBDBM10520(9-{[7-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)hept...)
Affinity DataKi: >1.00E+4nM ΔG°: >-28.5kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM10520(9-{[7-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)hept...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of fetal bovine serum AChE using acetylthiocholine iodide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed