Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50003024'
TargetAdenosine receptor A1(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  0.990nMAssay Description:Binding affinity towards adenosine A1 receptor in rat forebrain membranes using N6-[3H]cyclohexyladenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  0.990nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity carried out with [3H]cyclohexyladenosine in guinea pig forebrain membranes against adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]- CHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity against adenosine A1 receptor using N6-[3H]cyclohexyladenosine as radioligand in guinea pig forebrain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Guinea pig)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50003024(CHEMBL84363 | 8-Dicyclopropylmethyl-1,3-dipropyl-3...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards adenosine A1 receptor using N6-[3H]cyclohexyladenosine in guinea pig forebrain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed