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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50080545'
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50080545((2-Amino-6-benzyl-4,5,6,7-tetrahydro-thieno[2,3-c]...)
Affinity DataEC50: >2.00E+4nMAssay Description:Allosteric modulatory activity at human adenosine A1 receptor expressed in CHOk1 cells assessed as drug level causing half maximal allosteric effect ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50080545((2-Amino-6-benzyl-4,5,6,7-tetrahydro-thieno[2,3-c]...)
Affinity DataEC50:  1.13E+4nMAssay Description:Enhanced 0.5 nM [3H]-CCPA dissociation from adenosine A1 receptor of rat brain cortex membranes compared to 100 uM CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed