Affinity DataKi: 1.70nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in HEK293T cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15.5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in CHO-K1 cells assessed as reduction in cAMP level in presence of 0.1 uM adenosine by f...More data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 0.1 uM adenosineMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at adenosine 2A receptor (unknown origin) in presence of 1 uM adenosineMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 10 uM adenosineMore data for this Ligand-Target Pair
Affinity DataIC50: 143nMAssay Description:Antagonist activity at human adenosine 2A receptor expressed in CHO-K1 cells assessed as reduction in cAMP level in presence of 10 uM adenosine by fl...More data for this Ligand-Target Pair