Report error Found 20 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50085658'
Affinity DataIC50: 11nMAssay Description:Agonist activity at human Adenosine A3 receptor transfected in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production after 30 m...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from mouse A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibitory activity against Adenosine A3 receptor by inhibiting specific [3H](R)-PIA binding to rat testis membranesMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity in membrane of CHO cell stably expressing recombinant human Adenosine A3 receptor in the presence of GTPgammaS using [3H]8-ethyl-4-m...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to Adenosine receptor A3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to human adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Bnding affinity in membrane of CHO cell stably expressing recombinant human Adenosine A3 receptor using [3H]8-ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-te...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for human Adenosine A3 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from human A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity towards Adenosine A3 receptor (W243 mutant receptor)More data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Binding affinity towards human Adenosine A3 receptor wild typeMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Tested for the binding affinity of A3 receptor by displacing N6-[[125I]-4-amino-3-iodobenzyl]-adenosine-5''-N-methyluronamide from membranes of CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Displacement of [125I]- AB-MECA from rat adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Binding affinity to rat adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Inhibition of [125 I]-IABMECA binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 796nMAssay Description:Binding affinity towards Adenosine A3 receptor (H95A mutant receptor)More data for this Ligand-Target Pair
Affinity DataKi: 1.88E+4nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
