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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50335711'
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(CHEMBL1650355 | N-2,6-bis4-methoxyphenyl)pyrimidin...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(CHEMBL1650355 | N-2,6-bis4-methoxyphenyl)pyrimidin...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(CHEMBL1650355 | N-2,6-bis4-methoxyphenyl)pyrimidin...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cell membranes after 180 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(CHEMBL1650355 | N-2,6-bis4-methoxyphenyl)pyrimidin...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of CELT-228 from human adenosine A3 receptor expressed in human HeLa cells incubated for 30 mins by fluorescence polarization binding as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335711(CHEMBL1650355 | N-2,6-bis4-methoxyphenyl)pyrimidin...)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells incubated for 30 mins by fluorescence polarization binding as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed