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Found 2 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM19165'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM19165(3-phenyl-5H-indeno[1,2-c]pyridazine | Aza-heterocy...)
Affinity DataIC50:  3.10E+4nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM19165(3-phenyl-5H-indeno[1,2-c]pyridazine | Aza-heterocy...)
Affinity DataIC50: >1.00E+5nMpH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed