Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM10000'
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM10000((4-fluorophenyl)(6-methoxy-1-benzofuran-2-yl)pyrid...)
Affinity DataIC50:  0.740nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione [1beta-3H] as substrate incubated for 1 hrs by scintillation counting ana...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM10000((4-fluorophenyl)(6-methoxy-1-benzofuran-2-yl)pyrid...)
Affinity DataIC50:  44nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1,2,6,7-3H ]androstenedione / androstenedione during aromatization. Afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed