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Found 3 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50025155'
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025155(3-(4-Amino-phenyl)-3-methyl-pyrrolidine-2,5-dione ...)
Affinity DataKi:  800nMAssay Description:Inhibition of Cytochrome P450 19A1 against Androstenedione at 0.25 uM (Km=55 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025155(3-(4-Amino-phenyl)-3-methyl-pyrrolidine-2,5-dione ...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Cytochrome P450 19A1 against Androstenedione at 0.25 uM (Km=55 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025155(3-(4-Amino-phenyl)-3-methyl-pyrrolidine-2,5-dione ...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Cytochrome P450 19A1 against testosterone at 1.5 uM (Km=0.13 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed