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Found 2 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50322860'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50322860((R)-N-((R)-6-(3-((R)-3-hydroxypyrrolidin-1-yl)prop...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50322860((R)-N-((R)-6-(3-((R)-3-hydroxypyrrolidin-1-yl)prop...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human bradykinin B1 receptor assessed as inhibition of Lys-desArg9-BK-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed