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Found 2 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor' and Ligand = 'BDBM50293885'
TargetB2 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50293885(8-((3-chloro-5-(1-methyl-1H-imidazol-2-ylthio)pyri...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50293885(8-((3-chloro-5-(1-methyl-1H-imidazol-2-ylthio)pyri...)
Affinity DataIC50:  43nMAssay Description:Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed