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Found 6 Enz. Inhib. hit(s) with Target = 'Bifunctional protein GlmU' and Ligand = 'BDBM92474'
TargetBifunctional protein GlmU(Escherichia coli)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  7nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Haemophilus influenzae)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  23nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Streptococcus pneumoniae)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  1.50E+4nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Staphylococcus aureus)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50: >2.00E+5nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed