Found 2 Enz. Inhib. hit(s) with Target = 'Broad substrate specificity ATP-binding cassette transporter ABCG2' and Ligand = 'BDBM50563665'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universities Of Shandong
Curated by ChEMBL
Universities Of Shandong
Curated by ChEMBL
Affinity DataIC50: 748nMAssay Description:Reversal of BCRP-mediated multidrug resistance in human KBV cells assessed as mitoxantrone IC50 at 10 uM after 72 hrs in presence of mitoxantrone by ...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universities Of Shandong
Curated by ChEMBL
Universities Of Shandong
Curated by ChEMBL
Affinity DataIC50: 843nMAssay Description:Reversal of BCRP-mediated multidrug resistance in human KBV cells assessed as mitoxantrone IC50 at 5 uM after 72 hrs in presence of mitoxantrone by M...More data for this Ligand-Target Pair