Found 4 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50260068' 
Affinity DataKi: 2.10nMAssay Description:Compound dilution series were prepared in DMSO via a 3-fold serial dilution from 2.5 mM to 42 nM. Compounds were then diluted 6:100 in assay buffer (...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of His-tagged BRD4 bromodomain 1 (67 to 152 residues) (unknown origin) using acetyl-histone H4 as substrate after overnight incubation by ...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of His-tagged BRD4 bromodomain 1 (K57 to E168 residues) (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Compound dilution series were prepared in DMSO via a 3-fold serial dilution from 2.5 mM to 42 nM. Compounds were then diluted 6:100 in assay buffer (...More data for this Ligand-Target Pair
